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4,6-dimethyl-1-({1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyrimidin-2-one
3-ethyl-1-[(2-phenoxypyridin-3-yl)methyl]urea
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methoxy-2,2-dimethylpropan-1-one
4-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-(propan-2-yl)pyrimidine
3-[5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridazine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
(2S,4S)-4-amino-1-{[5-(2-cyanophenyl)furan-2-yl]methyl}-N-ethylpyrrolidine-2-carboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
1-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-6-methylquinolin-2-yl)piperidin-3-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
1-(2-ethoxyethyl)-2-oxo-N-(2,2,6,6-tetramethylpiperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N'-(2-methylphenyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanediamide
1-(3,5-difluorophenyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-cyclopropyl-1-{1-[4-(hydroxymethyl)benzoyl]piperidin-4-yl}piperidine-3-carboxamide
1-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-[1-(methoxymethyl)cyclobutanecarbonyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-chloro-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1H-indole-2-carboxamide
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}azocane
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[2-(2-methoxyphenoxy)ethyl]methylamine
2-[(4-benzylpiperazin-1-yl)methyl]-N-cyclopropyl-N-ethyl-1,3-oxazole-4-carboxamide
3-[(4-tert-butylphenyl)methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
methyl(oxolan-3-ylmethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-(carbamoylmethyl)-N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-fluoro-3-methylbenzoyl)piperidine
N-(3-methyl-1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
N'-(4-methylphenyl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]propanediamide
2-(methylsulfanyl)-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-[2-(3-methoxypropyl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
(2R,3R,6R)-3-phenyl-5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3,4-dimethoxyphenyl)-1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-(3-hydroxyphenyl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
5-(furan-3-yl)-1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
5-chloro-3-fluoro-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine
methyl 4-{[(2-oxopyrrolidin-3-yl)carbamoyl]amino}benzoate
1-{3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-3-phenylpropyl}-1H-1,2,4-triazole
N-[4-(furan-2-yl)butan-2-yl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[4-chloro-2-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenoxy]acetamide
3-(hydroxymethyl)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
1-(2-chloropyridin-3-yl)-3-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)urea
(4aR,7aS)-1-ethyl-4-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
3-(2-methoxyphenoxymethyl)-1-propyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-6-yl}-1H-1,2,4-triazole
1-[3-(3-methoxypropyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-benzyl-3-[(4-fluorophenyl)formamido]-N-(2-hydroxyethyl)propanamide
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})(1,3-thiazol-4-ylmethyl)amine