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N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[(dimethylcarbamoyl)amino]acetamide
4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)pyridine
1-cyclopentyl-N3-methyl-4-oxo-N5-(prop-2-en-1-yl)-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
6-[3-(ethylsulfanyl)phenyl]-3H-imidazo[4,5-b]pyridine
N-[3-(1H-imidazol-1-yl)butyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3,3-dimethyl-1-[(5-{[4-(propan-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
8-(2-amino-2-methylpropyl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aS,7aR)-5-methyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(5-ethylpyridin-2-yl)methyl]-N-methylpiperidine-2-carboxamide
3-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-(4-{4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}piperidin-1-yl)ethan-1-one
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
[(4-fluorophenyl)methyl]({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(cyclohexylmethyl)-5-[(2-methoxyethyl)(methyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(4-{[5-(2-cyanophenyl)furan-2-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
1-(2,3-dimethoxyphenyl)-2-(thiophen-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(3S,4R)-1-(3-chloro-5-methoxybenzoyl)-3-ethyl-4-methylpiperidin-4-ol
3-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}quinolin-7-ol
1-{4-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]thiophen-2-yl}ethan-1-one
2-(4-fluorophenoxymethyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrimidin-4-ol
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[(1-phenylcyclohexyl)formamido]methyl}benzoate
N,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)-5-propyl-1-benzofuran-2-carboxamide
4-(2,2-dimethylpropyl)-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
4-(2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperazin-2-one
N-{1-[1-(1-aminocyclobutanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
4-methyl-N-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)-1,2,3,6-tetrahydropyridine-1-carboxamide
1-(methoxymethyl)-N-[(3-phenylphenyl)methyl]cyclopropane-1-carboxamide
4-[1-(3-phenoxypropyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl]amine
ethyl 1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(5-ethoxyfuran-2-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-{1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}acetamide
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dimethoxybenzamide
4-methyl-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}-2-oxopentanamide
3-methyl-5-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(3-methylthiophen-2-yl)methyl]amino)ethan-1-ol
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]urea
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(5-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
2-(dimethylamino)-2-(4-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]acetamide
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
4-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1,2-dihydroquinolin-2-one
5-methyl-N-[1-(thiophen-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine