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N-{[1-(4-phenylbutanoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
4-{[3-(6-methoxypyridin-2-yl)phenyl]methyl}morpholine
(4aS,8aR)-6-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
3-benzyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
1-(2-{2-methyl-7-oxo-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-6-yl}ethyl)piperidine-3-carboxamide
3-(3-fluorophenyl)-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}benzamide
methyl 3-cyclobutaneamido-5-{[(2-methylphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(3-methoxyphenyl)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-{[1-(methylsulfanyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
1-benzyl-3-(2-methoxyphenyl)-6-(oxan-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-oxo-N-(2-phenylethyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
6-(methoxymethyl)-N-[(2,3,6-trifluorophenyl)methyl]pyridine-2-carboxamide
1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
3-(pentan-2-yl)-8-(3-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(3R,4R)-1-(2-ethylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-{[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzoic acid
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N-[(4-methoxyphenyl)methyl]-5-(3-methylbenzoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-amino-2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine-5-carbonitrile
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(morpholine-4-carbonyl)pyridin-2-amine
1,3,5-trimethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-4-sulfonamide
2-(1H-pyrazol-1-ylmethyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-oxazepane
7-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{5-[1-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-[(2-hydroxyethyl)(methyl)amino]benzamide
5-{[2-(dimethylamino)-2-(3-methylphenyl)acetamido]methyl}thiophene-2-carboxylic acid
2-(cyclopropylmethyl)-8-(2-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl (4aS,8aR)-6-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylate
4-{3-[(2-chlorophenyl)methyl]-1,2-oxazole-5-carbonyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
(2R)-2-amino-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
4-[(2-fluorophenyl)methyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-chlorophenyl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
N-[(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(1R,5R)-N,N-dimethyl-6-[3-(pyridin-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]propanamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-oxazole-4-carbonyl)piperidine
(1S,5R)-3-(morpholine-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-[(2,5-dimethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(4-fluoro-2-methoxyphenyl)-1-phenyl-1H-1,2,3,4-tetrazole
1-(4-chloro-3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)-1H-pyrazole
1-[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-2-yl)piperazine
ethyl 4-{[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]methyl}-1H-pyrazole-3-carboxylate
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide