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N-{2-[(2,5-dimethylthiophen-3-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
8-(5-chloropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[4-(4-cyanophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
3-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]ethan-1-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(3-phenylbutyl)(pyridin-4-ylmethyl)amine
N-{1-[1-(quinoxalin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}quinoline
N,4-dibenzyl-4-(hydroxymethyl)piperidine-1-carboxamide
{1-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-3-yl}methanol
(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
5-{imidazo[1,2-a]pyridin-6-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyridine
4-methyl-2-(propan-2-yl)-N-[1-(pyridin-4-yl)propyl]-1,3-thiazole-5-carboxamide
S-(4-fluoro-3-methylphenyl)-2-oxo-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}ethane-1-sulfonamido
N-({5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(4-hydroxybutyl)morpholine-2-carboxamide
1-(7-methyl-3-{[(2-phenylpropyl)amino]methyl}quinolin-2-yl)piperidin-4-ol
1-(2-cyclohexylethyl)-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-(3,4-difluorophenyl)-5-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
2-oxo-3-(pentan-3-yl)-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-ethyl-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-sulfamoylbenzamide
6-(2-methylpropyl)-2-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2-dihydropyrimidine-4-carboxamide
9-(dimethyl-1,2-oxazole-4-carbonyl)-1-methyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4,9-triazaspiro[5.5]undecane
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[2-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
(5S,9aS,9bS)-5-(2-chlorophenyl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(2-methoxyphenoxy)-1-(piperidin-3-ylmethyl)piperidine-4-carboxylic acid
3-[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]-N-(3-fluorophenyl)propanamide
3-(3-methoxypropyl)-1-[3-(2-methylphenyl)propanoyl]piperidine-3-carboxylic acid
4-fluoro-N-({1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}methyl)benzamide
1-(7-fluoroquinazolin-4-yl)-3-(2-methylphenyl)pyrrolidin-3-ol
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidine
(2S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-2-carboxamide
N-ethyl-4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylprop-2-en-1-yl)butanamide
7-cyclohexyl-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}cyclopentyl)pyrrolidine
3-(3-hydroxy-3-methylbutyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
2-cyclopropanecarbonyl-8-(4-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-fluoro-4-methyl-2-[2-(1,2-oxazolidine-2-carbonyl)pyrrolidin-1-yl]quinazoline
[(3R,4R)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-phenyl-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1H-1,2,3-triazole-5-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3-phenylpropyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepane