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2-[(1S,5R)-3-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
6-chloro-2-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N,N-dimethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
N-[2-({[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}amino)ethyl]acetamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-3-fluoro-4-methylbenzamide
N-ethyl-5-[7-methyl-4-(pyrrolidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-[(2E)-3-phenylprop-2-en-1-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-fluoro-N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-[(1-propyl-1H-imidazol-2-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
N-[(5-methylpyrazin-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(3S,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
4-(2-hydroxypyridine-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[2-(2,3,6-trimethylphenoxy)ethyl]acetamide
(4aR,8aR)-4-{[2-(trifluoromethyl)phenyl]methyl}-octahydro-2H-1,4-benzoxazine
1-(pyrrolidin-1-yl)-3-[1-(quinoline-6-carbonyl)piperidin-4-yl]propan-1-one
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-[2-(thiophen-2-yl)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxylic acid
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
N3-(3-methylbutyl)-N5-[(1-methylpiperidin-3-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[6-(propan-2-yl)pyridin-2-yl]piperazine
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyridin-3-yl)ethyl]pyridin-2-amine
2-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(4-{4-[3-(methoxymethyl)pyrrolidin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-yl)phenol
2-(3-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
4-chloro-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-5-methyl-1,3,4-oxadiazole
2-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
N-[(4-methoxyphenyl)methyl]-1-methyl-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(2-methoxyethyl)({[5-(methoxymethyl)furan-2-yl]methyl})({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)phenyl]acetamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-({1-[(4-ethylphenyl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
4-[(4-fluorophenyl)methyl]-1-(1,3-thiazol-2-ylmethyl)piperidine
2-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
7-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-ethyl-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
2-{2-chloro-4-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]phenoxy}acetic acid
(3S,4R)-4-(3-methoxyphenyl)-1-(1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
4-hydroxy-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidine-4-carboxylic acid
1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
N3-benzyl-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopentyl-5-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
1-(2-{1-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(1R,9aR)-1-[({2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
5-amino-3-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-(1-ethylpiperidin-4-yl)-4-(1H-pyrazole-3-carbonyl)-1,4-diazepane-6-carboxylic acid