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4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)butan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
3-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-6-ethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)acetamide
1-[(2-chloro-4-fluorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperidin-4-amine
(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[3-(cyclopropylmethyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
2-cyclopropyl-5-[(2S,5R)-2,5-dimethylpiperazine-1-carbonyl]pyrimidine
8-(cyclopropylmethyl)-N-[(4-fluorophenyl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
5-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(trifluoromethyl)pyridine
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(1-phenylethyl)-1H-1,2,3-triazole
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methylphenyl)ethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
3,3-dimethyl-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
benzyl 3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1'-(2-methoxypyridine-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-ethyl-5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-(propan-2-yl)-1H-pyrazole
1-[2-(2-methoxyethyl)piperidin-1-yl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-3-ol
3-(2-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
2-(dimethylamino)-N-(2-methanesulfonylethyl)-2-(2-methylphenyl)acetamide
N-[2-(morpholin-4-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[3-(1-methylcyclopropyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(4aS,7aR)-1-(4-methoxy-2-methylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-3-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(3-methoxypropyl)-1-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
7-methyl-3-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
(1S,5R)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N5-(3-methoxypropyl)-N6-[2-(1-methylpyrrolidin-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
5-(2-phenylphenyl)pyrimidine
N-{3-[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}acetamide
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
8-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{[3-(furan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
[(4-fluorophenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(4S,6R)-6-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-2-sulfanylidene-1,3-diazinane-4-carboxamide
6-(2,5-difluorobenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methyl-1,2-oxazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6,7-dimethoxy-2-[1-(oxan-4-yl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
2-cyclohexyl-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}pyrimidine
2-{3-[(3-carbamoylphenyl)methyl]pyrrolidin-1-yl}acetic acid
(5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}furan-2-yl)methanol
N,N-dimethyl-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1,2-oxazole
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[4-(pyridin-3-yloxy)piperidin-1-yl]ethan-1-one
[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine