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2-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)benzonitrile
methyl 3-benzamido-5-{[(4-acetamidophenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(thiophen-2-ylmethyl)piperidine
1-({3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}methyl)azepan-2-one
4-(furan-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
5-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrazin-2-ol
N-[2-(4-chlorophenyl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
8-(4-acetylbenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-benzyl-N-ethyl-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-methoxy-N-methylpyrimidin-4-amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
(2H-1,3-benzodioxol-5-ylmethyl)(methyl)({5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
4-fluoro-N-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)benzamide
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
1-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}piperidine-2-carboxamide
ethyl 1-benzyl-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[2-(pyridin-2-yl)ethyl]-4-(quinolin-5-yloxy)piperidine-4-carboxamide
N,N,4,5-tetramethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-2-amine
2-(2-phenyl-1H-imidazol-1-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-(pyridin-3-yl)-4-[(2,3,4-trifluorophenyl)methyl]piperazine
(1,4-dioxan-2-ylmethyl)({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(pyrimidin-4-ylmethyl)amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]propanamide
4-[4-(2-methoxyphenyl)piperidin-1-yl]pyrimidine
N-benzyl-3-hydroxy-N-(1,3-thiazol-2-ylmethyl)pyridine-2-carboxamide
2-methyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
7-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(6-aminopyridin-3-yl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}acetic acid
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-methylphenyl)methyl]amino}-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methoxyphenyl)acetamide
[(2,4-difluoro-3-methoxyphenyl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
{4-[1-cyclohexyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
3-methanesulfonamido-N-methyl-N-(oxan-2-ylmethyl)propanamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(1-hydroxypropan-2-yl)benzamide
1-(4-chlorophenyl)-4-(2-methoxy-4-methylbenzoyl)-5-methylpiperazin-2-one
1'-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
8-benzyl-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2-methylpyridin-3-yl)oxy]-1-(oxolane-2-carbonyl)piperidine-4-carboxylic acid
3-ethyl-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
4-(1,3-benzothiazol-2-yl)-2-{[(propan-2-yl)amino]methyl}phenol
3-[5-(1-ethylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
2-[(4-chlorophenyl)methyl]-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
5-methyl-2-(2-methylpropanamido)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
N,N-dimethyl-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]azepan-4-amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(dimethylamino)acetamide
2-{4-[(2,6-difluorophenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol