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1-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
5-(5-chloro-2-fluorophenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methylpiperidin-2-one
2-methoxy-N-[1-methyl-2-(pyridin-4-yl)-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
ethyl 3,5-dimethyl-4-{[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}-1H-pyrrole-2-carboxylate
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-amino-6-(6-methoxypyridin-3-yl)-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
N-[2-(pyrazin-2-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1,3-benzoxazole
4-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[2-(1H-1,2,4-triazol-1-yl)ethyl]amine
methyl 6-(3-methyl-2-oxopentanoyl)-2-{[(4-methylphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-(4-methyl-1H-pyrazol-3-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
3-[(4aR,7aS)-4-[(carboxymethyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
7-[methyl(1,3-thiazol-2-ylmethyl)sulfamoyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-(propan-2-yl)-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
(2S,4R)-4-[4-({[(3,4-dimethylphenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
4-methyl-7-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-2H-chromen-2-one
ethyl 4-benzyl-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylate
1-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)-4-phenylpiperazine
3-(4-fluoro-3-methylphenyl)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl 2-(2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)acetate
3-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(benzyl)(2-phenylethyl)amine
3-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]pyridin-2-ol
ethyl 3-[(3-chlorophenyl)methyl]-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
2-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}-4-methoxyphenol
{1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-3-(hydroxymethyl)piperidin-3-yl}methanol
4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
1-{[5-(1-ethylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpiperazine
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
1-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-methyl-3-(morpholin-4-yl)propan-1-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-(propan-2-yl)pyrimidin-2-amine
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
methyl 2-hydroxy-5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzoate
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-N'-(4-methylphenyl)propanediamide
3-(4-ethylphenyl)-N-methyl-N-[2-(methylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
(2S,4R)-4-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
(2,4,6-trimethyl-3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)methanol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one
2-[(1S,5R)-6-[(5-fluoro-2-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-{2-[(1-cyclopropyl-6-oxopiperidin-3-yl)formamido]ethyl}pyridine-3-carboxamide
methyl 4-[5-methyl-4-({4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)-1,3-oxazol-2-yl]benzoate