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N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-methylbenzene-1-sulfonamide
3-[2-(aminomethyl)-4-fluorophenyl]-N-ethylbenzamide
methyl 4-{[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]carbamoyl}piperazine-1-carboxylate
6-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-[6-(methoxymethyl)pyrimidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-4-(1H-pyrazol-3-yl)benzamide
N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
2-ethyl-8-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2-methoxyethyl)-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
8-[2-(2-chlorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1-methyl-1H-imidazol-2-yl)({1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl})methanol
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[(methylsulfanyl)methyl]piperidine
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]benzamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-methylpentanamide
N-(2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}ethyl)-3-methylpyridin-2-amine
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-fluoro-4-phenylbenzoyl)piperidine
N-(4-chloro-2,6-dimethylphenyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
2-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}({[4-(methylsulfanyl)phenyl]methyl})amino)ethan-1-ol
N-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)-N-(quinolin-6-yl)piperazine-1-carboxamide
2-methyl-N-[2-(pyridin-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
benzyl(methyl){[3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-oxazol-5-yl]methyl}amine
2-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperidine-3-carbonyl)pyridine
N,N,2-trimethyl-7-[3-(1H-pyrazol-1-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[5-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)furan-2-yl]benzonitrile
1-{4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-4-methylpentane-1,2-dione
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
5-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1H-1,2,3-benzotriazole
(4aS,8aR)-6-(2,3-difluorobenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
1-{[1-(2H-1,3-benzodioxol-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
3-(2-methylphenyl)-1-[2-(phenylamino)pyrimidine-5-carbonyl]pyrrolidin-3-ol
2-[(1R,5S)-3,6-diazabicyclo[3.2.2]nonan-6-ylmethyl]benzoic acid
(4aR,8aS)-N,N-dimethyl-1-{2-[4-(methylsulfanyl)phenyl]acetyl}-decahydro-1,6-naphthyridine-6-sulfonamide
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-2-[3-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
5-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
5-(2-hydroxybenzoyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-fluorophenyl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
1-methyl-6-oxo-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1,6-dihydropyridine-3-carboxamide
6-(3-chlorophenyl)-N,N-dimethylpyridine-2-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]oxane-2-carboxamide
2-[1-(4-aminopyridin-3-yl)-1H-pyrazol-4-yl]ethan-1-ol
N-ethyl-1-({4-[(5-methyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl}methyl)pyrrolidine-3-carboxamide
2-({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol