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N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-4-(methoxymethyl)benzamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl})amine
6-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
(4aR,8aR)-7-[(2-ethylphenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
2,6,8-trimethyl-4-(3-phenylpiperazine-1-carbonyl)quinoline
(3R,4R)-3-cyclopropyl-4-methyl-1-(pyrazine-2-carbonyl)pyrrolidin-3-ol
3-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-1H-pyrazol-5-amine
4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]benzene-1-sulfonamide
5-[1-(2-hydroxypyridine-3-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-4-yl)ethan-1-one
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxypropyl)acetamide
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
(4aS,8aR)-1-(3-aminopropyl)-6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(5-fluoro-2-methylphenyl)methyl]piperidine-4-carboxamide
(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]pyrrolidin-3-amine
4-benzyl-3-ethyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-5-one
[5-({3-[3-(dimethylamino)propoxy]phenyl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
3-{[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl](ethyl)amino}-1λ6-thiolane-1,1-dione
5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-oxazolidin-2-one
1-[2-(3-methylphenoxy)ethyl]-4-(pyrrolidin-1-yl)piperidine
N-cycloheptyl-N,6-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-(3-fluorophenyl)-3-[(2-oxopyrrolidin-3-yl)sulfamoyl]benzamide
N-[2-(furan-2-yl)ethyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-propylpiperazin-2-yl}ethan-1-ol
1-[(2-chlorophenyl)methyl]-N-[(3-methyloxetan-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-fluoro-N-{4-[4-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)piperidin-1-yl]phenyl}benzamide
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-2,5-dimethyl-1,3-thiazole
ethyl 1-(2-oxo-2-phenylacetyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
3-(dimethylamino)-N-[3-(2-methoxyphenyl)phenyl]piperidine-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-4-methylpentane-1,2-dione
1-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
1-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-{2-[3-(3-fluoro-4-methoxybenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
4-(8-methoxy-2-methylquinolin-5-yl)thiophene-2-carboxamide
6-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
2-(cyclopropylmethyl)-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-methoxy-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-phenylpyrrolidin-2-one
4-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-(2,5-dichlorophenyl)-3-methyl-5-(oxan-3-ylmethyl)-1H-1,2,4-triazole
1-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[3-(phenylsulfanyl)propyl]benzamide
4-[3-(pyrimidin-4-yl)piperidin-1-yl]pyrimidine
3-{2-[3-(ethoxycarbonyl)-3-(2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate