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1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
1-{2-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyrazin-2-yl)ethyl]amine
N-methyl-2-{4-[4-(1H-pyrazol-5-yl)phenyl]phenyl}acetamide
(3S,5R)-1-(2H-1,3-benzodioxole-5-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
(2E)-3-(3,4-difluorophenyl)-1-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
3-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-5,6-dihydro-1,4-dioxine-2-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
N-({1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
1-({3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
5-methyl-N-[(5-methylpyrazin-2-yl)methyl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
5-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3-phenyl-1,2,4-oxadiazole
N-(3-{6-[(2-hydroxyethyl)amino]pyridazin-3-yl}phenyl)acetamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-aminocyclopropanecarbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-3-carboxamide
3-(2-fluorophenyl)-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(diphenylmethyl)-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-6-(furan-2-yl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}thian-4-amine
1-cyclopropanecarbonyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-2-carboxamide
3-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]urea
1-benzoyl-N-[2-(2-fluorophenoxy)ethyl]piperidin-4-amine
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
2-[(propan-2-yl)amino]-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}pyrimidine-5-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-(thiophene-3-sulfonyl)piperidine-4-carboxylate
4-(1-{4-[6-(piperidin-1-yl)pyrimidin-4-yl]phenyl}ethyl)morpholine
9-(1,2,4-oxadiazol-3-ylmethyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[methyl({4-[3-(3-methylphenyl)piperidine-1-carbonyl]phenyl})amino]ethan-1-ol
1-methyl-2-oxo-N,3-diphenyl-1,8-diazaspiro[4.5]decane-8-carboxamide
methyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)azepan-2-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]benzamide
methyl[(2-phenyl-1,3-thiazol-5-yl)methyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
5-(1-benzyl-1H-pyrazol-4-yl)-3-(methoxymethyl)-1H-1,2,4-triazole
3-amino-N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}benzamide
2-chloro-4-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
2-{5-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-(2-fluorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(naphthalen-2-yloxy)propanamide
N-cyclohexyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(pyridin-2-ylmethyl)acetamide
9-ethyl-1-methyl-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[5-(2H-1,3-benzodioxol-5-yl)furan-2-carbonyl]morpholine
4-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}thiomorpholine
(1R,5S,8R)-8-methoxy-3-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-azabicyclo[3.2.1]octane