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(4aR,8aR)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-octahydro-2H-1,4-benzoxazine
6-[4-(piperidine-1-sulfonyl)phenyl]-3,4-dihydroquinazolin-4-one
2-amino-8-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-(cyclobutylmethyl)-2-[1-(2-fluorophenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
7-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-amino-6-(2,5-dimethoxyphenyl)-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-4-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}phenol
N-methyl-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-(quinoxalin-6-ylmethyl)propanamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-methoxypropanamide
(3aS,6aS)-2-[(3-fluoro-4-methylphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
3-(5-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazol-3-yl)pyridazine
1-[(2-chlorophenyl)methyl]-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1,4-dioxan-2-ylmethyl)[(3-fluoro-2-methylphenyl)methyl]methylamine
2-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenoxy)acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
(4aR,8aR)-1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
1-(4-{4-[1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenyl)ethan-1-one
2-(2-methoxyphenyl)-1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazole
5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]isoquinoline
5-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
5-{2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
[(2S,6S)-4-(5-ethyl-1,3-oxazole-4-carbonyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-(1-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzenesulfonamide
4-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-({[(2R)-1,1-diphenylpropan-2-yl]carbamoyl}methyl)piperidine-4-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-(cyclopropylmethyl)-4-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
4-methyl-2-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
[3-(cyclopropylmethyl)-1-(1,4-dithiepan-6-yl)piperidin-3-yl]methanol
5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1-(2-phenylethyl)-1H-1,2,4-triazole
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
N,1,3-trimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
3-benzyl-8-(1-methoxypropan-2-yl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(pyridin-3-yl)propanamide
ethyl 4-{2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
1-cyclopropyl-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
2-{5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-methyl-1H-1,3-benzodiazole
3-[3-({[2-(2-chlorophenoxy)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N-{2-[7-(2,2-dimethylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
2-ethyl-5-(3-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine