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2-(4-fluorophenyl)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]azetidine
dimethyl({3-[2-(quinolin-4-yl)-1H-imidazol-1-yl]propyl})amine
N-(oxan-3-yl)-1-oxo-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
(3ar,6ar)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-cycloheptyl-3,4-dihydropteridin-4-one
1-cyclopentyl-5-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrrolidine-3-carboxamide
3-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(2-methyl-5-sulfamoylphenyl)urea
ethyl 3-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole-2-carboxylate
7-methyl-2-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-hydroxy-2-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
4-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]-1-methanesulfonylpiperidine
1-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}piperidin-3-ol
4-(2,5-dihydro-1H-pyrrole-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-(3,4-dichlorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-({3-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
methyl 3-({[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate
4-{1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}benzonitrile
(3R,5S)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(naphthalen-2-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
7-(cyclohexylmethyl)-2-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(1-propylpyrrolidin-3-yl)acetamide
2-phenoxy-N-[1-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-ethyl-3-methoxy-N-(2-methylprop-2-en-1-yl)benzamide
6-(methylamino)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(propan-2-yl)-4-(pyridine-2-carbonyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
N-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
1-(3-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}phenyl)imidazolidin-2-one
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-ethyl-4-methyl-1,3-oxazole
4-{3-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}piperazin-2-one
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(4-{1H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetamide
4-[4-(dimethylamino)phenyl]-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-[ethyl(pyridin-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
methyl 3-{[(4-methyl-1,3-oxazol-5-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
1-{3-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-cyclopropyl-7-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[5-(methoxymethyl)thiophene-2-carbonyl]-1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](oxolan-2-ylmethyl)amine
N,3,6-trimethyl-N-(2-methylpropyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-N-(pyridin-4-ylmethyl)propanamide
(3R,4R)-1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-4-ethylpiperidine-3,4-diol
3-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
7-[3-(benzenesulfonyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-methyl-N-[(4-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(2,2-diphenylethyl)({3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine