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1-cyclopropyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
2-methyl-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]phenol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-N'-(2,4,6-trimethylphenyl)butanediamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-2-one
N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(trifluoromethyl)benzamide
2-(2-phenylethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-benzoxazole-5-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
7-chloro-3-{[(3-hydroxypropyl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
N'-cyclopentyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]butanediamide
1-(cyclohex-3-en-1-ylmethyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-(4-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
4-(3-aminopyrrolidine-1-carbonyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]benzene-1-sulfonamide
N-[2-(dimethylamino)ethyl]-2-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
N-methyl-N-(1-methylpiperidin-4-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N'-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-N,N-dimethylbutanediamide
3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
N-[(3S,4R)-1-[2-(3-methoxyphenyl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
N-(1H-indol-3-yl)-2-(methylsulfanyl)pyridine-3-carboxamide
1-[(2S)-oxolane-2-carbonyl]-3,3-diphenylpiperidine
8-{[3-(pyrimidin-4-yl)piperidin-1-yl]sulfonyl}quinoline
N,1-dimethyl-3-(propan-2-yl)-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazole-5-carboxamide
2-(5-methylfuran-2-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
(3aS,6aS)-2-[(3,4-difluorophenyl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
4-{1-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-3-methoxyphenol
3-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
3,5-difluoro-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylsulfanyl)acetamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]pyrazine-2-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-methyl-1H-pyrazole-3-carboxamide
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide
N-benzyl-N-butyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-methoxy-6-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
N-{2-[(7-fluoro-2-oxo-1,2-dihydroquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
(2S)-2-(methoxymethyl)-N-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]pyrrolidine-1-carboxamide
1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]-3-methylpiperidine-3-carboxylic acid
N-ethyl-N-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(3-methylpyridin-2-yl)ethyl]acetamide
N-[3-(1H-indol-4-yl)phenyl]acetamide
4-methyl-6-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyrimidin-2-amine
3-(4-methylphenyl)-N-{2-[3-(methylsulfanyl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
4-(2-fluorophenoxy)-1-(2-propoxypropanoyl)piperidine-4-carboxylic acid
4-{1-[2-(pyrrolidin-1-yl)pyrimidine-5-carbonyl]piperidin-4-yl}thiomorpholine
4-(2-methoxyethyl)-3-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole