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N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-3-yl)propanamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-[(dimethylamino)methyl]-N-[2-(ethanesulfonyl)ethyl]benzamide
6-{1-[3-(difluoromethoxy)benzoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
2-(dimethyl-1,2-oxazol-4-yl)-1-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N-[1-(2-methoxyethyl)-7-(3-oxopiperazine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
5-amino-3-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-[5-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
(2S)-2-{[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanamide
9-(3-hydroxybenzoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]benzamide
ethyl 1-(5-methoxyfuran-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
4-methyl-6-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-5-(prop-2-en-1-yl)pyrimidin-2-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(3-methoxyphenyl)acetamide
2-(2-methoxyethoxy)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
2-(4-ethylpiperazin-1-yl)-N-methyl-N-(oxan-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
1-methyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]azepane-2-carboxamide
7-[(4-aminoazepan-1-yl)sulfonyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
1-[2-(dimethylamino)ethyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]azepane
(2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[methyl(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
ethyl 2-[(5-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-amino-3-ethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-2-yl}pyridine
N-cyclopropyl-3-{5-[(3-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[(2,4-dimethoxyphenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}pyrrolidine-3-carboxylic acid
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-ethoxypyridine-3-carbonyl)pyrrolidin-3-yl]methanol
5-chloro-2-oxo-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-2-(methylamino)pyridine-4-carboxamide
1-[3-(1H-pyrazol-1-yl)phenyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
methyl 5-[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1,5-dimethyl-4-{[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1H-pyrrole-2-carbonitrile
N-(1,2-oxazol-3-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-[(3R,4S)-1-[(4-ethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1S,3R)-3-amino-N-[(3-chloro-2-fluorophenyl)methyl]cyclopentane-1-carboxamide
1-methyl-2-oxo-8-(quinolin-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4,6-dimethylpyridine-3-carbonitrile
1-(2-methyl-1-benzofuran-5-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
3-benzyl-4-{3-[(dimethylamino)methyl]benzoyl}piperazin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-({4-[4-(3-methylphenoxy)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
1-methyl-2-phenyl-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
N-{[7-(2-ethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-methylfuran-3-carboxamide