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7-[(3-methylphenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,4S)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-[(3R,4S)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(5S,9aS,9bS)-2-phenyl-5-(1-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 2-({4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidine-1-carbonyl}amino)acetate
2-butyl-N-[3-(methylsulfanyl)propyl]-1,3-benzoxazole-5-carboxamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
(4aR,7aS)-1-acetyl-4-(3,5-difluoropyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-{2-[(2-phenoxyethyl)amino]ethyl}pyrrolidin-2-one
[(3-methoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
8-cyclopropanecarbonyl-2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
3-(3-chlorophenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
[4-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](cyclohexyl)methanol
[(3R,4R)-1-(1,3-benzothiazol-2-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
3-chloro-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
1-(3-{[(2-chloro-4-fluorophenyl)carbamoyl]amino}propyl)piperidine-4-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]oxolane-2-carboxamide
N-{[(2S,4S)-4-fluoro-1-[2-(4-oxo-1,4-dihydroquinolin-1-yl)acetyl]pyrrolidin-2-yl]methyl}-2-methoxyacetamide
2-(2-hydroxyethyl)-9-[3-(3-methoxyphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[4-(oxan-2-ylmethoxy)phenyl]-1H-imidazol-2-yl}pyridine
N-methyl-6-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
3-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1-(4-methoxyphenyl)urea
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-butyl-5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
9-[3-(ethylsulfanyl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[(4-methoxy-3-methylphenyl)methyl]amino}-5-(methylsulfamoyl)-N-[3-(methylsulfanyl)phenyl]benzamide
5-fluoro-2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-cyano-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzene-1-sulfonamide
[1-(2-amino-5-ethylpyrimidin-4-yl)-3-[(dimethylamino)methyl]piperidin-3-yl]methanol
1-[3-(benzyloxy)phenyl]-3-[1-(2-hydroxyethyl)piperidin-4-yl]urea
3-(morpholin-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-(2-methoxyacetyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
2-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-phenylpiperidine-1-carboxamide
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-amine
N-{[2-(cyclopentyloxy)phenyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-(2-methylpropyl)-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2,5-dimethoxyphenyl)-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-({4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)quinoline
2-(6-aminopyridin-3-yl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
(4-{4-[(2-fluorophenyl)methoxy]benzoyl}-1,4-oxazepan-6-yl)methanol
1-phenyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide