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1-{4-[(3S)-3-hydroxypyrrolidin-1-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(propoxymethyl)pyrrolidin-1-yl]ethan-1-one
5-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
8-fluoro-N-methyl-N-(quinoxalin-6-ylmethyl)quinoline-2-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
3-(1H-imidazol-2-yl)-1-[(4-methylphenyl)methyl]urea
(4aR,8aR)-7-(5-acetylthiophene-2-carbonyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
5-hydroxy-1,2-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-3-carboxamide
4-[4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carbonyl]piperazine-1-sulfonamide
2-[5-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)furan-2-yl]benzonitrile
5,6,7-trimethoxy-N,N-dimethyl-3-[({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}amino)methyl]quinolin-2-amine
[(2R)-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-2-yl]methanol
5-fluoro-N4,N4-dimethyl-N2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidine-2,4-diamine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(2,4-dimethoxyphenyl)ethyl]-1,3-oxazole-4-carboxamide
2-({7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)-8-fluoroquinolin-4-ol
(1R,5R)-N,N-dimethyl-6-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3S,5R)-1-(3-fluoro-4-methylbenzoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(3aR,6aR)-2-[2-(5-acetylthiophen-3-yl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methoxy}phenyl)-1H-1,2,3,4-tetrazole
(1R,5R)-6-[(6-methylpyridin-2-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
5-benzyl-3-(pyridin-3-ylmethyl)-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(benzenesulfonyl)-2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrrole
3-methyl-1-(1-{6-[methyl(2-methylpropyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
1-[2-(dimethylamino)ethyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-methyl-8-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-methyl-3-(pyridin-2-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
methyl 1-{[(2-ethyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazole-3-carboxylate
5-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}pyrimidin-2-amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-amino-6-(4-fluorophenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5-methylpyridine-3-carbonitrile
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazine
[1-(thiophene-2-sulfonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
2-methyl-5-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3,4-thiadiazole
2-[(3-chlorophenyl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)morpholine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-(2-phenylethyl)-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[4-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)phenyl]acetamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
4-{[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-[(4-fluoro-2-methoxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
ethyl 2-(1-{1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-amido}cyclohexyl)acetate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-3-ol
N'-(3-ethylphenyl)-N-methyl-N-(pyrazin-2-ylmethyl)butanediamide
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-(2-phenylethyl)piperidine