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N-benzyl-N-butyl-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4,6-dimethyl-2-[3-methyl-4-(propan-2-yl)piperazin-1-yl]pyrimidine
{1-[2-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}methanamine
3-(pyrazin-2-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
3-{[1-(2-aminoethyl)-1H-1,2,3-triazol-4-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
1-[(2-ethylpyrimidin-5-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(1S,6R)-9-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpiperidine
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
N-(2-hydroxy-2-phenylethyl)-2-(2-methoxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-methyl-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-(2-methoxyethyl)-2-(1-methylpiperidin-2-yl)-N-(pyridin-3-ylmethyl)acetamide
5-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-1-[(2,4-difluorophenyl)methyl]azepan-2-one
1-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
N-(1,2-oxazol-3-ylmethyl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
4-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)-1-propylpyrrolidin-2-one
2-{4-[2-(thiophen-2-yl)ethyl]piperazin-1-yl}pyrazine
N-(5-fluoro-2-methylphenyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carboxamide
ethyl 1-benzoyl-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
3-ethyl-1-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]urea
2-{2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
8-methoxy-2-[(4-phenylpiperazin-1-yl)methyl]quinoline
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
8-(butan-2-yl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
{3-[(2,4-difluorophenyl)methyl]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl}methanol
2-phenyl-5-(2-propoxyethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl[(3-methylpyridin-4-yl)methyl]{[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
5-[1-(3-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydropyridin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}pent-4-enamide
1-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
3-(3-fluorophenyl)-4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-2-one
2-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
(3R,4S)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-amine
N-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
3-methoxy-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-{3-[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
4-(1H-1,2,4-triazol-5-ylmethyl)-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]urea
2-ethoxy-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
1-[(1S,2R)-2-butylcyclopropanecarbonyl]-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
3-(2-hydroxyphenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
3-propyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
3-(2-methoxyethyl)-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}piperidine-3-carboxylic acid
ethyl 1-(2H-1,3-benzodioxole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate