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(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3-benzyl-1H-1,2,4-triazol-5-yl)-4-(furan-2-carbonyl)piperazine-1-carboxamide
6-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(3R)-1-[(1-{[1-(2,4-dimethylbenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
3-[(2-ethoxyphenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
(1R,6S)-3-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
3,5-dimethyl-N-[2-(pyridin-4-yl)ethyl]-1-benzofuran-2-carboxamide
2-{2-[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}pyridine
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}phenyl)-2-(morpholin-3-yl)acetamide
1-(2-{4-[3-(2-methylphenyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
6-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(3aS,6aS)-2-acetyl-5-[(2-fluorophenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(3-methylphenyl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-[(4-fluorophenyl)methyl]-4-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]piperazin-2-one
1-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
(2R)-2-cyclohexyl-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-hydroxyethan-1-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-{[4-(hydroxymethyl)phenyl]methyl}urea
methyl 1-[(3R,5S)-1-[(4-ethylphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(2-fluorophenyl)-N-(1H-indol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
methyl (1R,3S,3aR,6aS)-3-(2-hydroxy-5-methylphenyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2S,4S)-4-amino-N,1-dimethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-N-methylpyrimidin-2-amine
3-[2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanamide
1-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
methyl 4-[(1R,9S)-5-amino-4-cyano-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-trien-3-yl]thiophene-2-carboxylate
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(phenylsulfanyl)acetamide
1-(4-{[5-(1,3-benzothiazol-2-yl)-2-hydroxyphenyl]methyl}piperazin-1-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
9-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
1-cyclobutanecarbonyl-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]piperidine-4-carboxamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)cyclopentane-1,3-dicarboxamide
N-{3-[4-({[4-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]phenyl}pyridine-4-carboxamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}[(4-ethylphenyl)methyl]methylamine
5-{4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}pyrazin-2-ol
methyl 1-(3-{4-[(cyclobutylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
4-(1,3-benzothiazol-2-yl)-2-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenol
1-(1,3,7-trimethyl-1H-indole-2-carbonyl)azepan-3-amine
N-methyl-2-(1-methylpiperidin-4-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3,7-dimethyl-11-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,7,11-triazaspiro[5.6]dodecane
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(morpholin-4-yl)ethan-1-one