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(2H-1,3-benzodioxol-4-ylmethyl)[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-(2-{4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-(2-hydroxyethyl)-2-methoxy-N-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-amino-4-{2-[3-(dimethylamino)propoxy]phenyl}-6-(furan-2-yl)pyridine-3-carbonitrile
4-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzonitrile
8-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(2-chloro-4-{[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
2-[(furan-3-ylmethyl)[(2-methylphenyl)methyl]amino]ethan-1-ol
2-(4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
ethyl 2-[({2-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-5-methoxyphenyl}methyl)(methyl)amino]acetate
2,3,5-trimethyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-oxopiperidin-3-yl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
[1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
3-chloro-N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyridine-4-carboxamide
N-[(4-fluorophenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
ethyl 1-[2-(4-benzamido-1H-pyrazol-1-yl)acetyl]piperidine-2-carboxylate
3-[({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-[2-(3-methoxyphenyl)-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
2-methoxy-5-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-{2-[2-(4-methylpentyl)morpholin-4-yl]-2-oxoethyl}piperidin-2-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-1,3-benzodiazol-1-yl)ethan-1-one
N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-(pyrazin-2-ylmethyl)acetamide
5-methoxy-N,1-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-indole-2-carboxamide
propan-2-yl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
[2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridin-4-yl]methanol
N-(1-{[(thiophen-3-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)benzamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-(1-propylpiperidin-4-yl)imidazolidine-2,4-dione
3-(3-fluoro-4-phenylbenzoyl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidine
[2-(1H-imidazol-1-yl)ethyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
9-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(2-chlorophenyl)-2-oxo-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]furan-3-carboxamide
1-(furan-2-ylmethyl)-3-(2-methoxyphenoxy)azetidine
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
6-oxo-2-(propan-2-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,6-dihydropyrimidine-5-carboxamide
(2S,4S)-4-amino-1-[4-(difluoromethoxy)benzoyl]pyrrolidine-2-carboxylic acid
7-(phenoxathiin-4-yl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,2-dimethyl-3-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propan-1-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
1-(4-methoxy-2-methylbenzoyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-chloro-4-{2-[(propan-2-yl)carbamoyl]phenyl}benzamide
5-[(2-fluorophenyl)methyl]-3-(3-methoxy-3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-{[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-ethyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
N,6,6-trimethyl-5-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}thiomorpholine-3-carboxamide
benzyl[(4-methyl-1,3-thiazol-5-yl)methyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
(3aS,6aS)-2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(thiophene-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid