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1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-amine
6-ethyl-2-methoxy-3-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3,7-dimethyl-11-[2-(propan-2-yl)pyrimidine-4-carbonyl]-3,7,11-triazaspiro[5.6]dodecane
ethyl 4-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazine-1-carboxylate
(2S,4S)-N-ethyl-4-(5-fluoro-2-methylbenzamido)-1-(4-methylpent-3-en-1-yl)pyrrolidine-2-carboxamide
1-(cyclobutylmethyl)-3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1-(oxolan-2-ylmethyl)urea
1-ethyl-N-(1-ethylpiperidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]acetamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-4-fluorobenzamide
2-(dimethylamino)-2-(2-methylphenyl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)acetamide
4-[(3-methylphenyl)sulfanyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-N-(5-methylpyridin-3-yl)benzamide
2-[4-benzyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N,N-dimethylacetamide
(cyclopentylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
4-benzyl-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)(methyl)[1-(pyridin-3-yl)ethyl]amine
N-{1-[1-(1H-imidazole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-(2-aminoethyl)-3-{methyl[(2E)-3-phenylprop-2-en-1-yl]sulfamoyl}benzamide
4-(furan-2-ylmethyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(3-chlorophenyl)methyl]pyrrolidin-3-yl}methyl)thiophene-3-carboxamide
N-{2-[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2-fluorobenzamide
3-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-3,4-dihydroquinoxaline-2-carboxamide
2-[4-chloro-2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenoxy]acetamide
3-[(benzylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
benzyl({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
5-ethyl-N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2,5,6-trimethylpyrimidine
5-[(benzyloxy)methyl]-1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazole
1-methyl-3-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indole
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
1-[2-(4-chlorophenyl)ethyl]-N-[(2-chlorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
1-methyl-2-(morpholin-4-yl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
2-(2H-1,3-benzodioxol-5-yl)-1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
(1R,6S)-N-butyl-6-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}cyclohex-3-ene-1-carboxamide
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-propyl-1,3-thiazole-4-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidine
6-ethyl-3-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-1,5-dimethyl-1,2-dihydropyridin-2-one
methyl 4-{5-chloro-2-[(1,3-thiazol-5-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-(3-methoxybenzoyl)piperazine
N,N-diethyl-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 4-[4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]benzoate
6-{3-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethylpyridazin-3-amine
N-methyl-N-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydronaphthalen-1-amine
methyl 4-({7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)benzoate
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](2-methoxyethyl)(oxolan-2-ylmethyl)amine