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N-[2-(furan-2-yl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
5-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-N-phenylpyridin-2-amine
N-(3,5-dimethoxyphenyl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-(3,3-diphenylpropyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
3-(1H-1,3-benzodiazol-2-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]propan-1-one
4-{[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]methyl}benzonitrile
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methylacetamide
4-[(4-fluorophenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(5-acetylthiophene-2-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
5-(4-fluorophenyl)-2-methyl-4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}pyrimidine
4-[3-(cyclobutylcarbamoyl)benzenesulfonyl]morpholine-2-carboxamide
N-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4,5-dimethylthiophen-2-yl)-2-methylpropanamide
4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)pyridine
2-(3-{1-[(3,4-dimethoxypyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-4-methylpiperidine
2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-8-methyl-2,8-diazaspiro[5.5]undecane
6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-9H-purin-2-amine
3-fluoro-4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1-[2-methoxy-5-({[2-(4-methoxyphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-(3-methyl-1-benzothiophen-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(4-tert-butylphenoxymethyl)-5-(3-methoxypiperidine-1-carbonyl)pyrimidin-4-ol
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(oxolane-3-carbonyl)piperidine
N-benzyl-N-[2-(dimethylamino)ethyl]-1-[1,3-dioxo-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}-N-cyclopentylbenzamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
(4aS,8aR)-6-(2-oxo-2-phenylacetyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-fluorophenyl)methyl]-3-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]propanamide
1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]-2-(pyridin-2-yl)ethan-1-one
1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)propan-1-one
1-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
(4aS,8aR)-6-(3-ethyl-1,2-oxazole-5-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
2-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
3-[5-(6-methylpyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-{1-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
2-(4-{4-[(2-phenylethyl)carbamoyl]phenoxy}piperidin-1-yl)acetic acid
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
1-[(2-aminopyridin-3-yl)methyl]-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid
4-(4-ethoxyphenyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-methyl-2-oxo-8-[4-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
N-cyclopropyl-2-({2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}formamido)acetamide
5,6-dimethyl-2-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}-2,3-dihydropyridazin-3-one