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(3S,4R)-3-benzyl-4-methyl-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-ol
N-(2-fluoroethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(1H-imidazol-1-yl)butan-2-yl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(5-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)-N-methylacetamide
N-cyclooctyl-5-[2-(hydroxymethyl)piperidine-1-carbonyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-(pyridin-2-yl)butyl]benzamide
ethyl 1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]piperidine-2-carboxylate
N-methyl-2-(4-phenylpiperidin-1-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-[(1-hydroxycyclohexyl)methyl]-3-(3-methanesulfonamidophenyl)urea
2-[(4-chlorophenyl)methyl]-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,3-benzoxazole
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3S,4R)-1-(furan-2-ylmethyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-(4-methoxy-3-methylphenyl)-5-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-butyl-11-{[2-(diethylamino)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-methoxy-2-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenol
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-ethyl-1H-pyrazole-3-carboxamide
[1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
5-(cyclopropylmethyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4R)-3-[ethyl({[1-(propan-2-yl)piperidin-4-yl]methyl})amino]-4-hydroxy-1λ6-thiolane-1,1-dione
N-(2-methoxyethyl)-3-(propan-2-yloxy)-N-(thiophen-2-ylmethyl)benzamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-phenylpiperidine-4-carbonitrile
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-cyclobutanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane
4-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-N-[3-(1H-imidazol-1-yl)propyl]pyridine-2-carboxamide
1-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)piperidine-3-carboxamide
2-[5-(oxolan-3-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
N-(3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropyl)-N-methylmethanesulfonamide
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
methyl 1-(benzyloxy)-8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(1-methyl-5-{[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
3-{1-[1-(2-methoxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
4-(2-{3-[(3-phenoxyazetidin-1-yl)methyl]phenoxy}ethyl)morpholine
4-[4-(4-acetylpiperazine-1-carbonyl)piperidin-1-yl]-2-[(2-chlorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
[2-(3-methoxyphenyl)-1-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]ethyl](methyl)(pyridin-2-ylmethyl)amine
(1S,2S)-2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)cyclohexan-1-ol
(3R,4S)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-propylpyrrolidin-3-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-methoxy-N-methyl-2-phenylacetamide
2-(2-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethoxy)ethan-1-ol
(1S,5R)-6-(5-chloro-2-fluorobenzoyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1,4-dithiepan-6-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[4-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
(4aS,7aR)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-2-methoxyphenol
N-(2-methylpropyl)-2-{9-oxo-4H,5H,6H,7H,8H,9H-[1,2,4]triazolo[3,2-b]quinazolin-2-yl}-N-(propan-2-yl)acetamide
6-methyl-2-(3-methylphenyl)pyridine-3-carboxamide