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7-methoxy-3-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
N-{[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}-3-(3-hydroxy-3-methylbutyl)benzamide
(3S)-N-tert-butyl-2-(5-hydroxypyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
7-(cyclopropylmethyl)-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-3,3-dimethylurea
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3R,4S)-1-(3-hydroxypropyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
methyl (2S,4R)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(4-phenylbenzamido)pyrrolidine-2-carboxylate
1-[3-(azepane-1-carbonyl)phenyl]-3-[1-(1H-imidazol-1-yl)butan-2-yl]urea
methyl 2-({3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}amino)benzoate
2-(4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(methylsulfanyl)benzamide
2-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]quinoline-2-carboxamide
5-[({1,9-dioxaspiro[5.5]undecan-4-yl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
N-{3-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]-2-methylphenyl}-2-methoxyacetamide
N-methyl-N-(2-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)methanesulfonamide
5-{1-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-cyclohexyl-4-{1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazin-2-one
6-[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,3S)-7-{[2-(benzylamino)pyrimidin-5-yl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
2-{[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
1-(3-methoxybenzoyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
N-ethyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}piperidin-3-ol
2-[1-(5-aminopyridin-3-yl)-1H-pyrazol-3-yl]-4-chlorophenol
2-[4-(1-methoxyethyl)phenyl]pyridine-4-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
5-fluoro-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1H-indole-2-carboxamide
1-ethyl-N-[1-(4-hydroxyphenyl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
{4-[(3-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
2-(2-methoxyethyl)-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
2-{4-[(3-fluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-4-carbonitrile
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[1'-(4-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
{1-ethyl-5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-{3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
6-chloro-2-methyl-N-[2-(propane-2-sulfonyl)ethyl]quinoline-4-carboxamide
8-methoxy-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]quinoline
(1S,5R)-3-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-cycloheptylpiperidin-3-yl)thiophene-3-carboxamide
1-[2-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)phenoxy]-3-[cyclohexyl(methyl)amino]propan-2-ol
1-[2-amino-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
[1-(2,3-dihydro-1H-indene-5-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
6-(benzyloxy)-1-(2-methylpropyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
[2-(8-methylquinolin-5-yl)pyridin-4-yl]methanol
N,N-dimethyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
1-cyclohexyl-4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
(1S,5R)-3-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one