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2-(cyclopropylmethyl)-N-(4-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[7-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
N-(1-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
(3R,5S)-N-[(2-ethoxypyridin-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-{2-[1-(2-ethoxybenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-ethyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-2-methylpyrimidin-4-amine
2-(5-chloro-2-methoxy-4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
(1S,4S)-5-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
1-cyclopentyl-4-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoyl)piperazin-2-one
6-methoxy-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(4,7-dimethylquinazolin-2-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(thiophen-3-yl)acetamide
4-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-4-acetamidobenzamide
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenylethan-1-one
2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
1-(4-methoxyphenyl)-3-methyl-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperazin-2-one
4-[5-(2-ethoxyethyl)-1,2,4-oxadiazol-3-yl]-1H-indole
8-fluoro-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}quinoline-2-carboxamide
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-3-phenyl-1H-pyrazole-4-carboxamide
1-[1-(4-fluorophenyl)propan-2-yl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(4aR,7aS)-1-(pyridin-3-ylmethyl)-4-(thiophen-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
3,5-dimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
methyl 6-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-3-(4-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
8-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(4-hydroxyphenyl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)propanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]methanol
2-(pyridin-4-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
7-(propan-2-yl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-(2,6-difluorophenoxymethyl)-N-[(2R)-2-hydroxypropyl]-1,2-oxazole-3-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
7-(1,3-benzothiazol-2-yl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N'-cyclooctyl-N-(2-hydroxy-2-phenylethyl)butanediamide
2-[2-(1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
N-cyclopropyl-6-methyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-N-(thiophen-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-fluoro-2-{4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperazin-1-yl}pyrimidine
5-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-methoxyphenol
1-({5-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-(3-chlorophenyl)-4-(1-methyl-2-oxoimidazolidine-4-carbonyl)piperazin-2-one
7-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]hex-5-enamide
(2S,4S)-4-amino-1-({[2-(4-chlorophenyl)ethyl]carbamoyl}methyl)-N-ethylpyrrolidine-2-carboxamide