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N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
2-hydroxy-N-[(4-methoxypyridin-2-yl)methyl]-4-(methylsulfanyl)butanamide
5-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
4-oxo-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
methyl 4-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-4-oxobutanoate
(3S,9aR)-8-(3-chlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(3-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}phenyl)amino]acetic acid
6-(2-chlorophenyl)-N-[2-(pyridin-3-yloxy)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-phenylpiperazine
3-(2-ethyl-1H-imidazol-1-yl)-N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}propanamide
N-[3-(3-fluorophenyl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)pyrrolidin-3-yl]acetamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
N-(4-fluorophenyl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-amine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-(1H-imidazol-2-yl)-N-methylbenzamide
methyl 2-[8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(1-benzylpiperidin-4-yl)-N,N-diethylpiperidine-3-carboxamide
(2S)-N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(pyridin-4-yl)piperazine
methyl 3-{[(2-cyclopropylquinolin-4-yl)formamido]methyl}-5-(pyrazine-2-amido)benzoate
N-[3-(2,5-dimethylphenoxy)propyl]-N-methyl-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
3-(2-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-(1H-pyrazol-4-yl)butan-1-one
2-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-3,5-dimethyl-1H-indole
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
N-[(2,3-dichlorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(2-hydroxyethyl)-6-methoxy-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
3-benzyl-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-5-carboxamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methanol
2-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]ethan-1-ol
N-ethyl-2-methyl-3-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)benzamide
N,N-dimethyl-4-[2-(4-methylpentyl)morpholine-4-carbonyl]piperidine-1-carboxamide
5-{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}-N-ethyl-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
1-{3-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-(1-benzofuran-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-[(4-methoxyphenyl)amino]-2-methylpropan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
8-fluoro-2-{[2-(pyridin-3-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
N4-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-6-ethyl-N2,N2-dimethylpyrimidine-2,4-diamine
[(5-ethylfuran-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-[(3,4-difluorophenyl)methyl]-8-[2-(oxolan-3-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole
2-hydroxy-4-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pentan-1-one