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1-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-1,4-diazepan-5-one
N-cyclopropyl-2-[3-(3-methoxypropyl)piperidin-1-yl]pyridine-4-carboxamide
3-ethyl-5-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-1,2-oxazole
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
8-[(2,3-difluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3-ethoxypropanamido)-N-(3-methoxyphenyl)benzamide
methyl 1-methyl-3-(3-phenylpropanamido)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
(5S)-5-[({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}but-2-yn-1-one
2-ethyl-5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrimidine
methyl 4-{[3-({[5-(methoxymethyl)furan-2-yl]formamido}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}benzoate
3-(1-methyl-1H-pyrazol-5-yl)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propan-1-one
4-(1-{4-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]phenyl}ethyl)morpholine
(4aS,8aR)-1-(3-aminopropyl)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-decahydro-1,6-naphthyridin-2-one
7-[(2,3-difluorophenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclohexyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
(3aR,7aS)-2-[(3,4-dimethoxypyridin-2-yl)methyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-ethyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-{[benzyl(methyl)amino]methyl}-N-(2,2-dimethylpropyl)-N-ethyl-1,2-oxazole-3-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-(thiophen-2-yl)butan-1-one
N-tert-butyl-7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidine
5,6,7-trimethoxy-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2-dihydroquinolin-2-one
1-[(2-ethoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-cyclopropyl-6-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,3-benzoxazole
1-[4-(4-fluorophenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
(4aS,8aR)-6-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
(2S)-1-[4-(adamantan-1-yl)piperazin-1-yl]-2-amino-3-(1H-imidazol-4-yl)propan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
[1-(1H-1,3-benzodiazol-2-yl)ethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-(1-methylpiperidin-4-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-indazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
(1S,5R)-3-(2,5-dimethylfuran-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
2-methyl-6-({4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-[(1S,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,4-dihydroquinolin-4-one
4-(1-phenyl-1H-pyrazol-4-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidin-2-amine
N-[(3S,4R)-4-(4-methylphenyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
N3-cycloheptyl-1-cyclopropyl-N5-[2-(2-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(1-benzylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
4-benzyl-3-ethyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepan-5-one
2-(3,4-dimethoxybenzenesulfonyl)-2,7-diazaspiro[4.5]decane
6-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]pyridine-2-carboxylic acid
4-(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
3-(2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanamide