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1-(4-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1S,6R)-3-(1H-indol-5-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-{[(4-methylphenyl)amino]methyl}benzamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-(propylcarbamoyl)pyrrolidine-2-carboxylate
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidin-3-ol
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-phenoxy-1-(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-1-yl)ethan-1-one
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
3-(furan-2-ylmethyl)-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-tert-butyl-4-{[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]methyl}furan-2-carboxamide
N-methyl-2-(morpholin-4-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-[1-(furan-2-carbonyl)pyrrolidin-2-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)thiophene-2-carboxamide
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-phenylpiperazine
1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidine
5-[1-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-1H-1,3-benzodiazole
2-(3-cyclopropyl-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazol-1-yl)benzoic acid
(1R,5R)-3-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(piperidin-1-yl)-3-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(4-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-ethyl-N-[(3-methoxyphenyl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(4aS,7aR)-1-(1-benzothiophen-2-ylmethyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-N-methyl-1-[(3-methylthiophen-2-yl)sulfonyl]pyrrolidine-2-carboxamide
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-N-(oxan-4-yl)propanamide
(4aS,8aR)-6-[(2,4-difluorophenyl)methyl]-1-methyl-decahydro-1,6-naphthyridine-4a-carboxylic acid
2,5-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-(3-hydroxypropyl)-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-(azepan-1-yl)-3-[3-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
1-(2-methoxyphenyl)-2,2-dimethyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-[1-(4-methanesulfonylphenyl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
4-({2-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
1-[4-(3-acetylphenyl)phenyl]-3-methyl-3-(1-methylpyrrolidin-3-yl)urea
(4aS,8aR)-6-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-amino-8-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(1-propyl-1H-1,2,3-benzotriazol-5-yl)-1H-pyrazol-1-yl]acetamide
3-(5-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
5-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide