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4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
2-benzoyl-8-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(2-methylphenyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(2,4-difluorobenzoyl)-3-(2-ethylphenoxy)azetidine
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-6-(2-methyl-1H-imidazol-1-yl)pyridazine
2-(2-oxopyrrolidin-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
(5S)-5-[({[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
N-(5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}thiophen-2-yl)acetamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine
1-[2-(1H-imidazol-4-yl)ethyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
2-(2H-1,3-benzodioxol-5-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazole
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}azepan-2-one
7-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
6-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile
methyl 3-[(3,5-dimethylphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
2-{4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}benzonitrile
5-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
1-[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-2-(morpholin-3-yl)acetamide
1-{4-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]piperidin-1-yl}ethan-1-one
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
2-{[4-amino-6-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)pyrimidin-2-yl]sulfanyl}-N,N-dimethylacetamide
1-[2-(dimethylamino)-4-[(pyridin-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-(2-methylpropyl)benzamide
5-(7-methoxy-4-methylquinolin-2-yl)pyridin-3-amine
3-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
5-methyl-6-(4-methylpiperidine-1-carbonyl)-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-(butan-2-yl)-1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
1-methyl-3-(pyridin-3-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-benzyl-1-[(4-fluorophenyl)methyl]-6-[3-(methylsulfanyl)propyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}piperazine
6-methyl-2-(pyridin-3-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrimidin-4-amine
methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
N-[(2-aminopyridin-3-yl)methyl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-[1-(4-amino-5-cyanopyrimidin-2-yl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-(4-chlorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide
3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-(1,2,3-thiadiazol-5-yl)urea
4-{[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-amine
ethyl 3-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butanoate
2-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
5-fluoro-2-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(pyridin-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-[(2,3-dimethoxyphenyl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-ethyl-2-{4-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenylacetyl]piperazin-1-yl}acetamide
1-[(1R,5S,6R)-6-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]butan-1-one
3-{2-[4-(3-methoxyphenyl)-3-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
1-{4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazin-1-yl}ethan-1-one