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N-[(2S)-pyrrolidin-2-ylmethyl]-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-[2-(pyridin-2-yl)ethyl]piperazine
4,6-dimethyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
N-methyl-7-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-phenoxyacetamide
14-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1,3-dimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
(4aS,7aR)-1-(pent-2-yn-1-yl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-(3-methylbutanoyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-3,4-dihydropyrimidin-4-one
(3S,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
2-(1-ethylpiperidin-4-yl)-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
3-methyl-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-3-phenylpiperidine
4-(benzyloxy)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidine
4-hydroxy-1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperidine-4-carboxylic acid
2-butyl-8-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-1-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}azetidin-3-yl)piperidine
4,6-dimethoxy-2-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
4-cyclohexyl-N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-oxopiperazine-1-carboxamide
3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)urea
(1R,3S)-3-(2-hydroxyethoxy)-7-(1H-1,2,3-triazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-(1-ethylpiperidin-4-yl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]ethan-1-one
3-{2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-methyl-5-[1-(3-phenylpropyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
3-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
8-chloro-N-[cyclopropyl(pyridin-2-yl)methyl]-N-methylquinoline-2-carboxamide
N-[(3-methylphenyl)methyl]-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
2-(adamantan-1-yl)-1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}ethan-1-one
1-{[(3-cyanophenyl)carbamoyl]amino}-N-methylcyclohexane-1-carboxamide
2-(dimethylamino)-4-methyl-N-[2-(pyridin-4-yl)ethyl]pyrimidine-5-carboxamide
3,4,7-trimethyl-N-(2-oxoazepan-3-yl)-1H-indole-2-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indol-3-yl)acetamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-cyclopropyl-3-{1-[3-(4-fluorophenyl)benzoyl]piperidin-3-yl}propanamide
1-cyclopropanecarbonyl-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
N2,N2,N4,N4-tetramethyl-7-[2-(methylamino)pyrimidine-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-({4-[(1,4-dimethyl-1H-pyrazol-5-yl)carbamoyl]phenyl}methyl)-N-ethylpyrrolidine-3-carboxamide
3-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}butanoic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
7-chloro-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
methyl 5-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-5-oxopentanoate
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-(oxan-4-yl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide