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N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methoxy-2-phenylacetamide
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-(4-hydroxy-3-methylbenzoyl)pyrrolidine-2-carboxamide
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
[(4-methanesulfonylphenyl)methyl](methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
4-benzyl-3-ethyl-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1,4-diazepan-5-one
2-[1-(carboxymethyl)-2-methyl-1H-indol-3-yl]-1H-1,3-benzodiazole-6-carboxylic acid
(1R,6S)-9-methyl-3-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
ethyl 4-(2-phenylethyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-4-carboxylate
(1R,5R)-3-[3-(difluoromethoxy)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(5-ethylfuran-2-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
N-ethyl-2-hydroxy-4-methoxy-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
(2S,4R)-4-amino-1-(4-acetamidobenzenesulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
methyl 1-[(3S,5S)-1-(1-benzylpiperidin-4-yl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-(1-methyl-1H-imidazol-2-yl)-1-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}-1H-1,2,3-triazole
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(3-methoxypyrazin-2-yl)-7-azaspiro[3.5]nonan-1-ol
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl](1,3-thiazol-2-ylmethyl)amine
3-{2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
methyl[(1-methyl-1H-pyrazol-4-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
5-(2,3-difluorophenyl)pyridine-2-carbonitrile
2-(azepan-1-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-{1-[1-(2,3-difluoro-4-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
6-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-2-carbonitrile
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
methyl 6-cyclobutanecarbonyl-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-({1-[(5-ethylthiophen-2-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(piperidin-1-yl)-3-[2-(pyridin-4-yl)phenoxy]propan-2-ol
3-(1-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1,2-dihydroquinolin-2-one
N-(3-aminopropyl)-1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(methylsulfanyl)-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2-ethoxyphenyl)methanol
2-[methyl({4-methyl-5-[1-(pyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
5-phenyl-N-(pyridin-2-ylmethyl)-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(3aS,6aS)-2-[(5-chloro-2-fluorophenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(benzyloxy)phenyl]-4-butyl-3-oxopiperazine-1-carboxamide
1-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
3-(2-{[(2,4-dimethoxyphenyl)methyl]carbamoyl}ethyl)-N,N-dimethylpiperidine-1-carboxamide
3-({2-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(furan-2-ylmethyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
13-[4-ethoxy-3-(hydroxymethyl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-fluoro-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
3-{methyl[2-(1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}-N-(2-methylbutyl)benzamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(1-{4-[(cyclobutylmethyl)(oxolan-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide