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8-(1H-1,3-benzodiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-[(4-fluorophenyl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(1-benzothiophen-2-ylmethyl)-N-methyl-2-(methylamino)pyridine-3-carboxamide
8-[(2R)-2-aminopropanoyl]-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-benzyl-2-(4-methyl-1,4-diazepan-1-yl)-N-[(3-methylpyridin-2-yl)methyl]acetamide
2-ethyl-1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(4-fluorobenzoyl)-decahydro-1,6-naphthyridin-2-one
1-{3,5-dimethyl-4-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
2-[4-(3-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
7-(2-ethylpyrimidine-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
3-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}pyridine
N-[(3R,4R)-3-hydroxy-1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl]pyridine-2-carboxamide
1-(3-methylfuran-2-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[4-(1,3-oxazol-5-yl)benzoyl]piperidin-3-yl]methanol
1-[1'-(cyclohex-3-ene-1-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]-3-(thiophen-3-yl)propan-1-one
3-(benzylamino)-N-cyclopentyl-5-(phenylsulfamoyl)benzamide
N-(5-methyl-1,2-oxazol-3-yl)-2-[3-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]-2-oxoacetamide
(1S,6R)-9-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-N-(3-methoxypropyl)-6-methylquinazolin-4-amine
6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,N-dimethylpyrazin-2-amine
methyl 3-(7-chloro-2-{[(2S)-2-acetamido-4-(methylsulfanyl)butanamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
1-[(4-methanesulfonylphenyl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-[(2,5-difluorophenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[3-(2,6-dimethoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
(2R,3S,6R)-3-(4-fluorophenyl)-5-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
4-methoxy-2-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
ethyl 4-[6-(2,4-dimethylbenzoyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
N-(2-hydroxyethyl)-5-(2-methoxyphenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(4-chlorophenoxy)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidine-4-carboxylic acid
(3R,5R)-N-(2-methylpropyl)-1-(pyridin-4-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
(2R)-2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4,4-dimethylpentan-1-one
N-methyl-2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethane-1-sulfonamide
methyl 3-(furan-3-amido)-5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4S)-1-benzyl-N-methyl-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
4-{3-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzoyl}morpholine
1-{1'-[(5-fluoro-2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-[bis(prop-2-en-1-yl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-(3-phenylpropyl)propanamide
1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
3-(2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1,2-oxazole-3-carboxamide
6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(3-methylbutyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide