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2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(furan-2-yl)-2-hydroxyethyl]acetamide
(4aS,8aR)-1-(2-aminoethyl)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[1'-(pyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[(3-methoxyphenyl)methyl]piperidine
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(1,2,5-thiadiazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2-amino-1,3-thiazol-4-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
2-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperidin-4-yl}-N-methylacetamide
2-methyl-3-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-indole
1-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
(2R,3R)-3-[methyl(quinolin-6-ylmethyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-cyclopentyl-5-(dimethyl-1,2-oxazole-4-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 3-[(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)amino]-4-methoxybenzoate
2-(thiophen-3-ylmethyl)-4-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-4-(oxan-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-fluoro-5-{3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
3-(4-methoxyphenyl)-4-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-pyrazole
6-(methoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]pyrimidin-4-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
N-[1-(pyrazin-2-yl)piperidin-4-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-{[1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-4-yl]methyl}acetamide
5-(oxane-4-carbonyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[(3-chlorophenyl)methyl]-N-(1H-imidazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-methyl-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-(naphthalen-2-yl)-1,2,4-triazine
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-1-(4-benzylpiperazin-1-yl)propan-1-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
9-[2-(4-ethylphenyl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyethyl)-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
(2S,4R)-4-amino-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
4-{5-[(dimethylamino)methyl]pyridin-2-yl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[3-(3-methylphenoxy)azetidine-1-carbonyl]pyridin-3-ol
7-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
6-(1-{[(1-cyclopentyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N,N-dimethylpyridine-3-carboxamide
1-[(2,4-difluorophenyl)methyl]-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}azepan-2-one
6-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]pyridine-3-carbonitrile
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
(2-{[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
7-(cyclobutylmethyl)-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
9-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}-4,6-dimethyl-2-(propan-2-yl)pyrimidine
(2S)-1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]pyrrolidine-2-carboxamide
1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-ol