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[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
2-{1-[(4-fluorophenyl)methyl]-4-(quinolin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[3-(1H-indol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
3-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-methyl-N-(pyridin-4-ylmethyl)-5-({[4-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenoxy)piperidine
1-(5-fluoro-2-methoxyphenyl)-3-[(3-methyloxetan-3-yl)methyl]urea
ethyl 1-[7-chloro-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)quinolin-2-yl]piperidine-3-carboxylate
2-(2-methylpentanoyl)-N-(2H-1,2,3,4-tetrazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
methyl 3-[(3,5-dimethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4R)-1-(2,3-difluoro-6-methoxybenzoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
(1S,2S)-2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)cyclohexan-1-ol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(4-ethylphenyl)methyl]-N-methylpropanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
N-methyl-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,6-dihydropyrimidine-5-carboxamide
2,6,8-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]quinoline
2-(1H-imidazol-2-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]benzamide
1-{1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzonitrile
5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
2-(cyclopropylmethyl)-8-(4,6-dihydroxypyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-imidazole
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-methyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]pyrrolidine-2-carboxamide
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-cyclopentyl-4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}benzamide
2-{[7-(1,3-benzoxazol-2-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
2-[4-(pyridin-4-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(4-methoxyphenyl)propanoyl]piperidine-3-carboxylate
2-(4-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
6-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-N-(9H-fluoren-9-yl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,3S)-3-methyl-2-{[1-(4-methylphenyl)propan-2-yl]amino}pentan-1-ol
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
2-(1-methyl-1H-indol-3-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-[2-(4-chlorophenyl)ethyl]-1,1-dioxo-N-(pyridin-3-ylmethyl)-1λ6-thiolane-3-carboxamide
(3S,4S)-1-(5-chloropyridine-3-carbonyl)-4-methylpiperidine-3,4-diol
1-(2-fluorophenyl)-2,2-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]cyclopropane-1-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-3-(pyrrolidine-1-carbonyl)-1,2-oxazole
1'-(isoquinolin-1-yl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(benzyloxy)methyl]-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-2-yl}pyridine
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
1-{4-[(2,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
(1s,4s)-N1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]cyclohexane-1,4-diamine
N-[(3S,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one