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(2S)-2-acetamido-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
1-cycloheptyl-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
5-(1-butyl-1H-1,2,4-triazol-5-yl)-N,N-dimethylpyridin-2-amine
methyl 1-[2-hydroxy-3-(4-{[(3-phenylpropyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
benzyl(cyclopropylmethyl){[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
3-{1-[2-(3-fluorophenyl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-methoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}butanamide
(1S,5R)-6-benzyl-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
3-cyano-N-(2-ethoxyphenyl)piperidine-1-carboxamide
N-[(2-fluorophenyl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
8-methoxy-2-methyl-5-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]quinoline
1-(3,5-dimethyl-4-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]propan-1-one
5-(2-methylpropyl)-1'-(5-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
(4S)-3,3,4-trimethyl-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol
6-(2-chlorophenyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}pyridine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
2-[4-(2-methoxyethoxy)phenyl]-6-methylpyridine-3-carboxamide
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrimidin-2-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(dimethyl-1,3-thiazol-4-yl)-N-methylacetamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(3-methylpiperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
3-chloro-N-cyclopentyl-4-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
8-fluoro-4-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydroquinoline-3-carboxamide
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]methyl}-4-methoxyphenol
2-(2,5-dimethoxyphenyl)-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-cyclohexyl-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
3-({1-[2-(2,3,4-trifluorophenyl)acetyl]pyrrolidin-3-yl}methyl)benzamide
ethyl 4-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-(cyclohexylmethyl)-N5-[(4-methoxyphenyl)methyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
6-(2-chlorophenyl)-N-[2-(dimethylamino)ethyl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(4-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}thiophen-2-yl)ethan-1-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(pyridazin-3-yl)pyrrolidin-3-yl]methanol
N-[(2-fluorophenyl)methyl]-2-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}acetamide
N-cyclopropyl-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyrrolidin-3-yl)benzamide
N-({8-[(3-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
(2E)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-3-(pyridin-2-yl)prop-2-enamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-{2-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-[2-(2,4-difluorophenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
1-{4-methyl-2-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidin-5-yl}ethan-1-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-3-phenyl-1,2-oxazole