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4-methyl-2-{2-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]ethyl}-1,3-thiazole-5-carboxylic acid
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-benzoxepine-4-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}thiomorpholine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazine
2-chloro-3-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
methyl 8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[2-(diethylamino)ethyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methylacetamide
1-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2-hydroxyacetyl)piperidin-3-yl]propan-1-one
N-[2-(furan-2-yl)ethyl]-3-[(1-methylpyrrolidin-3-yl)sulfamoyl]benzamide
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
(2S,4R)-4-amino-N-ethyl-1-(4-methanesulfonylbenzoyl)pyrrolidine-2-carboxamide
N-[(2R,3R)-2-ethoxy-1'-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N,4-dimethyl-5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
3-{[1-(ethylcarbamoyl)pyrrolidin-3-yl]methyl}benzoic acid
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(3-phenoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N4-(3,3,3-trifluoropropyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-(1,3-benzoxazol-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-cyclohexyl-4-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)benzamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(pyridin-3-yloxy)ethyl]benzamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[(3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-ethoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-(1-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
N-cyclopropyl-2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-4-carboxamide
4-(2-methylpropyl)-1-(3,4,5-trifluorobenzoyl)-1,4-diazepan-5-one
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)naphthalene-1-sulfonamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
1-[2-(1-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-1H-indazole-3-carboxylic acid
5-(3-acetylphenoxymethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-ethyl-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
1,3-dimethyl-5-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-1H-pyrazolo[3,4-d][1,3]thiazole
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-({[5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-ylmethyl]-6-methylquinolin-4-ol
2-{1-[(2-methylphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(furan-2-yl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azepane
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(2,3-difluorophenyl)methyl]pyrrolidin-2-one
2-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}-N,N-dimethylethane-1-sulfonamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-benzyl-3-fluoro-N-(3-hydroxy-2-methylpropyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-ethynylbenzamide
1-(3-methylcinnolin-5-yl)-3-[2-(3-phenylpyrrolidin-1-yl)ethyl]urea