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2-(azepan-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-amino-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
1-[(2-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
2-amino-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-fluoro-2-methyl-N-(propan-2-yl)quinoline-4-carboxamide
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)piperidin-2-one
1-{4-[2-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-oxoethyl]phenyl}imidazolidin-2-one
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
1-[2-(1H-imidazol-1-yl)ethyl]-4-({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperazine
3-methyl-5-(5-methyl-1,2-oxazol-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
4-(2H-1,3-benzodioxol-5-yl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(furan-2-yl)-1-(oxane-4-carbonyl)azepane
3-phenyl-1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperidine
5-methyl-3-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}-1H-indole-2-carboxylic acid
[(3R,4R)-1-(3-ethoxybenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[(3-phenyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-2-yl)piperidin-4-ol
N-({5-[(2,2-dimethyloxan-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-4-phenylbutane-1,2-dione
3-ethyl-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-{4-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]piperidin-1-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[2-(morpholin-4-yl)acetyl]pyrrolidine-3-carboxylic acid
N-methyl-N-(pyrazin-2-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-cyclopropyl-5-methyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
3-{1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(6-chloropyridin-3-yl)-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
(1R,5R)-6-benzyl-3-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-({2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)phenoxy]ethan-1-ol
6-[(2S,5R)-2,5-dimethylpiperazin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(2S,4R)-N,N-diethyl-4-[2-(1H-indol-1-yl)acetamido]-1-methylpyrrolidine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
methyl 3-[(4-methoxyphenyl)methyl]-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-methyl-4-[2-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]piperazine
N,N-dimethyl-5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}furan-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(furan-3-ylmethyl)piperidine
6-(2-ethoxybenzoyl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1,3-dimethyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(methoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]cyclobutane-1-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1S,5R)-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-2,1-benzoxazole
[(5-ethylpyridin-2-yl)methyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
1-[(5-methylfuran-2-yl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
5-(4-methoxyphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-oxo-1-phenylpyrrolidine-3-carboxamide
N,2-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
5-{[benzyl(methyl)amino]methyl}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide