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1-methyl-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(naphthalen-2-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-acetylbenzamide
3-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-(1-methylpiperidin-4-yl)-2-[(phenylsulfanyl)methyl]-3,4-dihydropyrimidin-4-one
3-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]propane-1,2-diol
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-yl)ethan-1-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-{[5-(furan-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}thiomorpholine
N-[2-(2,3-dimethoxyphenyl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(1R,5S)-N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-1-methyl-1H-pyrrole-2-carboxamide
2-(benzyloxy)-N-{[(2S,4S)-4-fluoro-1-(2-methylfuran-3-carbonyl)pyrrolidin-2-yl]methyl}acetamide
1-cyclopentyl-3-methyl-5-[5-(oxan-2-yl)furan-2-yl]-1H,4H-pyrazolo[3,4-d]imidazole
N-cyclopropyl-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydroquinoline-4-carboxamide
4-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(4,7-dimethylquinazolin-2-yl)-N-[2-(3-fluorophenyl)ethyl]piperidine-4-carboxamide
N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-(thiophen-2-ylmethyl)acetamide
2-{2-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
N-[2-(dimethylamino)-1-phenylethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
6-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1H-indene-5-carboxamide
2-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
1-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]butan-2-ol
{3-[(3-chlorophenyl)methyl]-1-(naphthalene-1-sulfonyl)piperidin-3-yl}methanol
3-cyclopentyl-1-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)urea
5-(4-fluorophenyl)-N-[2-(1H-imidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-amido}piperidine-1-carboxylate
6-(2-methoxyethyl)-2-(3-{[methyl(oxan-4-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-[5-(furan-3-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
methyl 3-[(3S,4R)-1-[(4-ethoxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
3-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
3-{5-[1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H-1,2,3-triazol-4-yl]thiophen-2-yl}prop-2-yn-1-ol
(5S,9aS,9bS)-2-cyclopentyl-5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 2-[butyl(methyl)sulfamoyl]-6-(2,3-dihydro-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1-benzothiophene-5-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-(oxan-2-ylmethoxy)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
N-cyclopropyl-1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)cyclohexanecarboxamide
2-{4-[2-(pyridin-4-ylsulfanyl)acetyl]morpholin-3-yl}acetamide
3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide