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2-methyl-3-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-{[5-(2,6-dimethylhept-5-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
3-{5-[6-oxo-1-(prop-2-en-1-yl)piperidine-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-ethyl-3-(piperidin-4-ylmethyl)-1-(1,3-thiazol-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-propyl-1,2,4-oxadiazole
3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-[3-(dimethylamino)propyl]propanamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-{[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
methyl 4-(4-{[6-(dimethylamino)pyridin-3-yl]methyl}piperazin-1-yl)benzoate
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
(1R,5S)-3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-3-propylpiperidin-3-yl]methanol
8-(2-fluoro-6-methoxybenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
5-(3,5-difluoro-4-methoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
3-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-6-fluoroquinolin-4-ol
6,7-dimethoxy-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1-[(4-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
3-butanamido-4-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
(3S,4S)-1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-(5-cyano-4,6-dimethylpyridin-2-yl)-1,4-diazepane-6-carboxylic acid
2-benzyl-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
[(3R,5R)-5-[(dimethylamino)methyl]-1-(1-phenylcyclopentanecarbonyl)piperidin-3-yl]methanol
N-cyclopentyl-2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(piperidin-3-yl)benzamide
2-[4-(dimethylamino)phenyl]-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
1-[(3-chlorophenyl)methyl]-N-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N,1-dimethyl-3-(propan-2-yl)-N-(quinoxalin-6-ylmethyl)-1H-pyrazole-5-carboxamide
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperidine-1-carboxamide
4-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}-6-methoxypyrimidine
methyl 4-(2-amino-5-butyl-6-methylpyrimidin-4-yl)piperazine-1-carboxylate
5-({[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}methyl)-2-methoxybenzoic acid
2-(2-ethoxypyridin-3-yl)-1,3-benzothiazole
methyl 3-({methyl[1-(methylcarbamoyl)ethyl]amino}methyl)benzoate
2-amino-3-ethyl-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-(propan-2-yl)acetamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
N-(3,5-dichlorophenyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-(1-ethylpiperidine-2-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
methyl 5-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-(2-chlorophenyl)-7-(prop-2-en-1-yl)-2-(thiomorpholine-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)cyclobutanecarboxamide
3-(furan-2-yl)-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
6-methoxy-N-(2-methoxyethyl)-2-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-3-carboxamide
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione