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2-{4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}phenol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-2-oxoimidazolidine-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N,N-diethyl-3-hydroxypiperidine-1-carboxamide
2-phenyl-4-[3-(pyridin-4-yl)azetidin-1-yl]quinazoline
N-(oxolan-2-ylmethyl)-2-(1H-1,2,4-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
9-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(piperidin-4-ylmethyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]benzamide
2,6-dimethoxy-3-[4-(1,3-oxazol-5-yl)phenyl]pyridine
2-{4-[(1-ethyl-1H-indol-3-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
4-ethyl-1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}ethan-1-one
ethyl 1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyrrolidin-1-yl)piperidine
8-[(2-aminopyridin-3-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(2-ethoxyethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
6-({[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}methyl)pyrimidin-4-ol
3-{2-[(5-ethylpyrimidin-2-yl)amino]ethyl}-1,3-oxazinan-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(piperidin-3-yl)piperidine-4-carboxamide
2-[(5-ethylfuran-2-yl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-amine
N-[(4-methoxypyridin-2-yl)methyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
methyl 5-{[1-(4-fluorophenyl)propan-2-yl]amino}-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(dimethylamino)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
{imidazo[1,2-a]pyrimidin-2-ylmethyl}({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
(1S,4S)-2-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-2,5-diazabicyclo[2.2.1]heptane
4-{4-[1-(2-chloro-4-methylphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-(3-methoxyphenyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-pyrazole-5-carboxamide
N-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
4-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methoxyphenol
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-2-(propan-2-yl)pyrimidine-5-carboxamide
2-(9H-fluoren-2-ylmethyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-2-(methylamino)benzamide
(1R,5R)-6-(cyclopropylmethyl)-3-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 5-{[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]methyl}-1-(2-methylphenyl)-1H-pyrazole-4-carboxylate
4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1-(propan-2-yl)piperidine
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-{1'-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl]propanoic acid
3-methyl-7-(4-phenoxybutyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 3-(cyclobutylmethoxy)-5-{[(3-methyloxetan-3-yl)methyl]carbamoyl}benzoate
(1R,5R)-6-(cyclobutylmethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-4-(3-fluorophenyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-tert-butyl-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
1-{[1-(hydroxymethyl)cyclobutyl]methyl}-5-methyl-5-phenylpiperidin-2-one
N-{1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide