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3-(4-benzylpiperazine-1-carbonyl)-2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-1,4-dihydropyridin-4-one
6-oxo-N-[2-(thiophen-2-yl)ethyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
1-(2,2-dimethylpropyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-ethyl-2-[4-(2-methylpyridin-4-yl)piperazin-1-yl]pyridine-3-carboxamide
2-(3-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
5-{[cyclopropyl({[4-(methylsulfanyl)phenyl]methyl})carbamoyl]amino}-2-fluoro-N-methylbenzamide
4-fluoro-3-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}benzene-1-sulfonamide
N4-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrimidine-2,4-diamine
1-[2-(morpholin-4-yl)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-fluoro-5-({[(2S)-1-hydroxy-3-phenylpropan-2-yl]carbamoyl}amino)phenyl]-2-methylpropanamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)benzamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
1-(4-chlorophenyl)-4-(3,5-difluoropyridine-2-carbonyl)-5-methylpiperazin-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1,4-dithiepan-6-amine
ethyl 1-({1-[(2-fluorophenyl)methyl]-7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperidine-4-carboxylate
8-cyclopropanecarbonyl-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-(4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}phenyl)methanesulfonamide
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-3-carboxamide
N-benzyl-3-[(cyclopentylamino)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
7-(cyclobutylmethyl)-2-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
7-(3,4-dihydronaphthalen-2-yl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
benzyl[(6-methylpyridin-2-yl)methyl](1,3-thiazol-2-ylmethyl)amine
5-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3,4,7-trimethyl-1H-indole-2-carboxamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
(3aR,6aR)-2-(2-methoxyethyl)-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(hydroxymethyl)-N-[3-(4-methylbenzenesulfonamido)propyl]-1H-1,3-benzodiazole-5-carboxamide
3-amino-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
3-(1-ethyl-1H-imidazol-2-yl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
3-benzoyl-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N,5-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl 4-[3-({[(4-fluorophenyl)methyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
4-cyclobutanecarbonyl-2-(4-methylpentyl)morpholine
(1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
N-[1-(3,5-difluorophenyl)cyclopropyl]-3-(1H-pyrazol-1-yl)benzamide
8-(1,3,7-trimethyl-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(8-methoxy-2H-chromen-3-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
methyl 6-{[benzyl(methyl)amino]methyl}-3-(2,5-dimethylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
[(3R,4R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-(4-methylphenyl)furan-2-carboxamide
3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1H-indazole
1-[(5-acetylthiophen-3-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[2-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
(3R,7S,8aS)-7-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(5-acetylthiophen-3-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-(2-oxoimidazolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide