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1-tert-butyl-5-cyclobutyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazole
4-(hydroxymethyl)-4-(oxan-2-ylmethyl)-N-(2-phenylethyl)piperidine-1-carboxamide
1-(5-chloro-3-fluoropyridin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-1-(piperidin-4-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-[1-(furan-3-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
6-methyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(2S)-1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-4-oxo-N-(propan-2-yl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-{4-[(2-chloro-5-fluorophenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
(3S)-2-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-N-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-methoxy-6-(3-{1-[3-(pyridin-3-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyridazine
methyl 3-cyclohexanecarbonyl-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(oxolane-2-carbonyl)piperidine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanoic acid
1-{4-[4-(2,6-dimethylquinoline-3-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
N-{2-[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
N-(pyridin-2-ylmethyl)-1-[1-(4,4,4-trifluorobutyl)piperidin-4-yl]piperidine-3-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1-[(3S,4R)-1-[(2-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-[1-(3-methylbut-2-en-1-yl)-4-(quinolin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]urea
2-phenoxy-N-(1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2,3-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-cyclobutyl-6-methyl-N-(oxan-4-ylmethyl)pyrimidin-2-amine
6-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
9-methoxy-N-methyl-7-oxo-3-{[4-(propan-2-yloxy)phenyl]methyl}-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(2-hydroxyethyl)({3-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl})amino]ethan-1-ol
N-ethyl-5-methyl-N-(2-methylprop-2-en-1-yl)-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-methoxy-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
2-amino-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
2-{[2-(diethylamino)ethyl]amino}-N-(2,4-dimethylphenyl)acetamide
3-methyl-2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1H-indole
2-(3-fluorobenzenesulfonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazine
[4-(2-phenylethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl]methanol
N-(furan-2-ylmethyl)-4-methyl-N-(prop-2-en-1-yl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7,8-dimethyl-3-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydroquinazolin-4-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N,1-dimethyl-3-propyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-5-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-(2-hydroxyethyl)pyrrolidine-3-carboxylic acid
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
1-[4-(4-chlorophenyl)piperazin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
methyl 1-ethyl-3-(oxolane-3-amido)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-6-methylpyridine