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3-{2-[5-(6-fluoro-1H-1,3-benzodiazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
1-ethyl-4-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-(1,4-dioxan-2-ylmethyl)-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
5-cyclopropanecarbonyl-1'-(oxolane-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-ethyl-1H-imidazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
1-[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
N-(2-methylpropyl)-1-[1-(propan-2-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-cyclopropyl-4-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrrolidin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
(1R,3R,5S)-8-(furan-2-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
1-(2,5-dimethoxybenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
(1-methyl-5-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-{1-[(2-cyanophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[(5-chloro-1-benzothiophen-3-yl)methyl]-4H-1,2,4-triazole
1-(3-cyano-4-methylphenyl)-3-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}urea
4-(1H-imidazol-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
6-fluoro-2-(pyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2-methyl-1,3-thiazol-5-yl)methyl]amine
N-[2-(3-methylthiophen-2-yl)ethyl]morpholine-2-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[(2-methylphenyl)methoxy]azetidine
1-(5-chloropyridin-2-yl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-cyclopropyl-2-fluoro-5-sulfamoyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
5-chloro-1,3-dimethyl-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-1H-pyrazole
N-[(8-methoxy-2H-chromen-3-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-3-amine
[(1r,4r)-4-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}cyclohexyl]methanol
4-methoxy-2-[(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
5-ethyl-2-methyl-4-[4-(2-phenylethyl)piperazin-1-yl]pyrimidine
N-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]piperidin-4-yl}methanesulfonamide
1-(2-methoxypyrimidine-5-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
6-fluoro-2-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}methyl)quinolin-4-ol
1-(3-chlorophenyl)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
6-ethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(morpholin-4-yl)pyrimidin-4-amine
5-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-3-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)benzamide
9-[(5-tert-butyl-2-hydroxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-ethyl-4-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
5-chloro-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
5-methyl-1-({3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[methyl(1-methylpiperidin-4-yl)amino]-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
(1S,5R)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[1'-(1H-indole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(2S,4S)-4-(3-methoxypropanamido)-N,1-dimethyl-N-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
4-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]benzamide
5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-cyclopentyl-N-methyl-6-oxo-N-(quinolin-2-ylmethyl)piperidine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-5-fluoropyridine-3-carboxamide