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5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
methyl[3-(5-methylfuran-2-yl)butyl](1,2-oxazol-3-ylmethyl)amine
(3aR,5S,6S,7aS)-2-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydro-1H-isoindole-5,6-diol
1-{2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-phenoxy-N-({7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
(3S)-3-benzyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-[3-(methylsulfanyl)propyl]urea
1-{6-[4-(1-methoxyethyl)phenyl]pyridin-2-yl}piperazine
1-(azocan-1-yl)-3-[4-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1,6-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-chloro-4-hydroxy-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}benzamide
1-{3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}azepan-4-amine
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
5-{[3-(morpholin-4-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-(2-methyl-4-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-1-(1-methyl-1H-imidazol-2-yl)ethan-1-ol
methyl 4-{4-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]piperazin-1-yl}benzoate
(1S,5R)-3-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
N-methyl-4-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}benzamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-7-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
1-amino-N-[(1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]cyclobutane-1-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)propanamide
9-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}-N,N-dimethyl-3-azaspiro[5.5]undecane-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[1-(2-acetylbenzoyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
N-(2-amino-4-methyl-1,3-benzothiazol-6-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
4-({5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
1-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)urea
N-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3-phenyl-1H-pyrazole-4-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-ol
1-methyl-2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
methyl 3-(4-fluorobenzenesulfonamido)-5-{[2-(thiophen-2-yl)acetamido]methyl}benzoate
4-{5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2-methoxyphenyl}morpholine
N-(4-cyclopentylpyrimidin-2-yl)-1-(propane-1-sulfonyl)azepan-3-amine
2-[4-(3-cyclopentylpropyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
N-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]morpholine-2-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(4-methylpiperazin-1-yl)ethan-1-one
N-[(3,5-difluorophenyl)methyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-[4-(thiophene-2-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
1-cyclohexyl-4-[6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carbonyl]piperazin-2-one
3-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-[(4-methylphenyl)methyl]propanamide