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4-(1,4-dimethyl-1H-indazol-3-yl)benzamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
(2-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
3-{[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl](methyl)amino}-1-phenylpropan-1-ol
8-fluoro-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]quinoline-2-carboxamide
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-methoxypyridine
4-[(4-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(dimethylamino)azepan-1-yl]propan-1-one
[5-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
3-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
N,N-dimethyl-2-{[2-(1H-pyrazol-1-yl)butanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(3-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propyl)-1H-1,2,3-benzotriazole
5-(methoxymethyl)-N-methyl-N-[1-(pyridin-2-yl)propyl]furan-2-carboxamide
3-propyl-6-[(3,4,5-trimethoxyphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(4-methyl-3-phenylpiperazin-1-yl)propan-1-one
6-(pyrrolidin-1-ylmethyl)-4-(quinoline-3-carbonyl)-1,4-oxazepan-6-ol
N-[2-(1H-indol-3-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
10-methoxy-5-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2,2-diphenylethyl)acetamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyrrolidin-3-yl)ethan-1-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(2-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
N-[(2-chloro-6-fluorophenyl)methyl]-N,2-dicyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N,N-diethyl-1-{[7-fluoro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidine-3-carboxamide
[(3-fluorophenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
2-{[9-(2-ethylbutanoyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzonitrile
1-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
2-[4-(pyrimidin-2-yl)piperazin-1-yl]-1-[2-(thiophen-2-yl)azetidin-1-yl]ethan-1-one
2-chloro-5-acetamido-N-(3-hydroxypropyl)-N-(thiophen-2-ylmethyl)benzamide
2-(3-hydroxyadamantan-1-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
3-phenyl-1-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)propan-1-ol
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]oxy}benzamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-1-(1H-pyrazol-1-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropane-1-carboxamide
2-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
6-(4-fluoro-2-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-(methylsulfanyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(2,5-dimethoxyphenyl)-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
1-{2-[2-(methylsulfanyl)phenyl]pyrimidin-4-yl}piperidin-3-ol
4-(2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-2-yl}ethyl)morpholine
5-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1'-[3-(1-phenylethyl)-1,2-oxazole-5-carbonyl]spiro[indene-1,4'-piperidine]
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-(4-chlorophenyl)-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(furan-2-yl)-2-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]propanoic acid
4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one