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1-[5-(1H-1,3-benzodiazol-1-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
N-(2-ethyl-6-methylphenyl)-3-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)propanamide
{7-[2-(propan-2-yloxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-[2-(4-methoxyphenyl)phenyl]-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-4-(4-methoxyphenyl)butane-1,4-dione
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidine
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(2-phenoxyethyl)piperazine
7-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[4-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]but-3-yn-1-ol
ethyl 2-(N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamido)acetate
3-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(furan-3-carbonyl)piperidine-4-carboxylic acid
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-(3-methoxyphenyl)acetamide
N-[(3-fluorophenyl)methyl]-4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]benzamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-(pyridin-4-ylmethyl)piperazin-1-yl]ethan-1-one
2-amino-4-ethyl-N-[1-(furan-2-carbonyl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-4-propylpyrimidine-5-carboxamide
5-{5-[(1-ethylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)spiro[azepane-4,2'-chromene]
2-chloro-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-5-(trifluoromethyl)benzamide
7-ethyl-2-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
6-(3-hydroxyazetidin-1-yl)-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
5-{[2-(1-ethylpiperidin-4-yl)acetamido]methyl}-N-methylfuran-2-carboxamide
4-{1-[4-(4-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
4-{1-ethyl-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-3-yl}benzamide
6-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-9H-purine
4-(azepane-1-sulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide
8-(2,4-dimethylpyrimidine-5-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
6-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,6-dihydropyridine-2-carboxamide
3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
N-[2-(4-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]pyridine-4-carboxamide
5-(oxolane-3-carbonyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
ethyl 2-{1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
(2H-1,3-benzodioxol-5-ylmethyl)[(3,5-dichloropyridin-4-yl)methyl](pyridin-3-ylmethyl)amine
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
4-methyl-2-(propan-2-yl)-6-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
1-(morpholin-4-yl)-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}propan-1-one
5-(2,4-difluorophenoxymethyl)-N-(1,3-dihydroxy-2-methylpropan-2-yl)-1,2-oxazole-3-carboxamide
5-methoxy-1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-indole-2-carboxamide
4-(1,3-benzothiazole-6-carbonyl)-1-methylpiperazin-2-one
ethyl 4-benzyl-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidine-4-carboxylate
N,6-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
1-(2-ethoxyphenyl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
1-{2-[3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione