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N-{3-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-3-oxopropyl}acetamide
2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}acetic acid
2-{4-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
N-(1-benzyl-1H-pyrazol-3-yl)-2-(1H-pyrazol-1-yl)acetamide
2-(3-hydroxyphenyl)-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
2-{4-[1-(1-cyclopropanecarbonylpiperidin-3-yl)-1H-1,2,3-triazol-4-yl]phenoxy}pyrimidine
2-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)acetamide
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-1-(piperidin-1-yl)ethan-1-one
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(2-methyl-1-benzofuran-5-yl)urea
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3,3-dimethylbutan-1-one
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
(4aR,7aS)-1-ethyl-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-cyclobutaneamido-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}benzamide
N-(adamantan-2-yl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(3-methoxypropyl)piperidine
3-[2-(dimethylamino)ethyl]-1-(6-fluoropyridin-3-yl)-3-methylurea
{1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-[(4-chlorophenyl)methyl]piperidin-4-yl}methanol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,1-dioxo-1λ6-thiane-4-carboxamide
2-(2-methoxyphenyl)-2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
methyl 4-({[2-(1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)ethyl]amino}methyl)benzoate
(3S,4S)-4-[methyl(2-methylpropyl)amino]-1-(4-phenyl-1H-imidazole-5-carbonyl)pyrrolidin-3-ol
7-chloro-1-(prop-2-yn-1-yl)-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-pyrrole-2-carboxamide
3-[2-(dimethylamino)ethyl]-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1-{[2-(furan-2-yl)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-(3-ethoxypropyl)-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1,9-dimethyl-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
[(1R,3S,3aS,6aR)-5-methyl-1-(2-methylpropyl)-3-[4-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-(4-methoxy-2-methylphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
N-tert-butyl-4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
dimethyl[({3-methyl-7-[4-(piperidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)sulfamoyl]amine
N-(3-hydroxypropyl)-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1-benzofuran-5-carboxamide
4-(5-fluoro-1-methyl-1H-indazol-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
ethyl 1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
methyl 3-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]carbamoyl}propanoate
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](ethyl)(pyridin-4-ylmethyl)amine
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]butanamide
({4-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
3-({2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}methyl)-5-(propan-2-yl)-1,2,4-oxadiazole
5-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
[(2,2-dimethyl-1-phenylcyclopropyl)methyl]({[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})methylamine
N-benzyl-1-(2-hydroxyethyl)-5-({4-[methyl(phenyl)amino]phenyl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(carbamoylmethyl)-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{5-[(2E)-pent-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-amine
(4-{[1-(1-benzofuran-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]thian-4-amine
[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-(4-{[3-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-(1-methyl-1H-imidazol-2-yl)-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)piperidine