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N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopentanecarboxamide
9-(4-methylpyrimidine-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclopropylmethyl)-N-methyl-5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(phenoxymethyl)-1H-pyrazole
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-(6-hydroxypyrimidin-4-yl)-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-diazepan-6-ol
3-(2-ethylbutyl)-8-(pyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(thiophene-2-sulfonamido)acetamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-{1-[(4-methylphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}butanamide
6-{4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
3-(1H-1,3-benzodiazol-2-yl)-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
8-methyl-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
(2R,3S,6R)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-hydroxyethan-1-one
ethyl 4-{[(trimethyl-1H-pyrazol-4-yl)carbamoyl]amino}piperidine-1-carboxylate
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
4-amino-N-ethyl-N-{[4-(propan-2-yl)phenyl]methyl}pyridine-2-carboxamide
4-fluorophenyl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
methyl 5-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-{[2-(propylamino)pyrimidin-5-yl]methyl}morpholine-2-carboxamide
3-{[2-(1-methyl-1H-pyrazol-5-yl)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
ethyl 5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[6-(4-cyclopentyl-1,4-diazepan-1-yl)pyrimidin-4-yl]piperidin-4-ol
N'-(4-butanamido-3-methoxyphenyl)-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
1-methyl-N-{1-[(3-methylphenyl)methyl]cyclopropyl}azepane-2-carboxamide
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
4-chloro-N,1-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
4-benzyl-3-[1-(1-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)-1,4-oxazepan-6-ol
3-(1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}piperidin-3-yl)benzoic acid
N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-benzyl-N-[(2,5-difluorophenyl)methyl]-1,3-thiazole-4-carboxamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl](3-phenylpropyl)amine
3-(2-{2-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(4-chlorophenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(thian-4-yl)piperazine-1-carboxamide
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-11-methyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-{[cyclohexyl(methyl)amino]methyl}-2-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
N-benzyl-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine