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2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
methyl 1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperidine-4-carboxylate
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(6-fluoroquinolin-2-yl)methyl]methylamine
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(propan-2-yl)pyrimidine-5-carboxamide
{1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-methyl-1-oxobutan-2-yl}urea
1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-2-(2-chloro-6-fluorophenyl)ethan-1-one
1-(2-methyl-1-benzofuran-7-carbonyl)-3-(piperidin-1-ylmethyl)piperidine
2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[2-(trifluoromethoxy)phenyl]methyl}acetamide
(3S,4R)-4-(3-methoxyphenyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
methyl 1-(3-{4-[(4-acetylpiperazin-1-yl)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-(4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-(furan-2-ylmethyl)-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
(2S)-3-(4-hydroxyphenyl)-2-(oxan-4-ylformamido)propanamide
(2S,4R)-4-amino-1-[(2-tert-butylpyrimidin-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-methyl-6-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzothiazol-2-amine
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-(1H-pyrazol-4-yl)butan-1-one
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-2-{4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]morpholin-3-yl}acetamide
4-(1H-imidazol-2-yl)-1-[3-(pyrrolidin-3-yl)benzoyl]piperidine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(pyridin-3-yl)ethyl]propanamide
methyl(1,2-oxazol-3-ylmethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl}methanesulfonamide
(4aS,7aR)-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-fluorophenyl)methyl]-N-methylacetamide
3-(2-methoxyphenyl)-5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
6-(furan-3-yl)-2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-{[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}-3-(furan-2-yl)propanoic acid
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(2-benzamido-5-methylphenyl)-1-(carbamoylmethyl)piperidine-4-carboxamide
(1R,3S)-3-(2-phenylpyrrolidine-1-carbonyl)cyclopentane-1-carboxylic acid
N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
ethyl 5-[2-(4-fluorophenyl)-3-oxopiperazine-1-carbonyl]-1H-imidazole-4-carboxylate
4-hydroxy-1-methyl-N-[2-(2-phenoxyphenyl)ethyl]piperidine-4-carboxamide
N-(pyridin-3-yl)-3-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzamide
4-(4-chlorophenoxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
3-(azocane-1-sulfonyl)-N-(1,2-oxazol-3-ylmethyl)benzamide
N-(2-hydroxyethyl)-3-(1H-imidazol-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-methylpiperidine
N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
4-({4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}methyl)-1H-indole
3-(3-methoxypropyl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
N-[1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidine
3-chloro-6-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-2-carboxylic acid