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5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
(3aR,7aS)-2-(2-methoxypyrimidine-5-carbonyl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2,2-dimethyl-N-(1-{1-[1-(5-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
4-amino-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
N-[(2R,3R)-1'-[(3,4-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
5-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzothiadiazole
3-(cyclopropylmethyl)-1-(3-methylbut-2-enoyl)piperidine-3-carboxylic acid
[1-(6-methylquinoline-4-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
N-(2H-1,3-benzodioxol-5-yl)-8-methyl-2-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}quinazolin-4-amine
2-(6-phenylpyridazin-3-yl)-2,8-diazaspiro[4.5]decane
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methoxy-3-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3,4-dichlorophenyl)-4-(2-methoxypyrimidine-5-carbonyl)morpholine
N-methyl-N-[2-(morpholin-4-yl)propyl]-2-propylpentanamide
(2R,3R)-3-amino-1'-[5-(trifluoromethyl)pyridin-2-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2,5-dimethyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]furan-3-carboxamide
4-{5-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-pyrazol-3-yl}phenol
1-{4-[(2,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(pyridin-4-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]propanamide
(2R)-2-hydroxy-1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-phenylethan-1-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(oxan-4-yl)benzamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-[4-(1H-imidazol-1-yl)phenyl]-N-[(2-methoxyphenyl)methyl]-N-methylpiperidin-4-amine
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-[2-(dimethylamino)ethyl]-5-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
(3S,9aR)-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-N-(1-{1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3-(hydroxymethyl)pyrrolidin-3-ol
1-(1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}azetidin-3-yl)piperidine
2-(adamantan-1-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(propan-2-yloxy)ethyl]amine
2-methoxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4-(piperidin-1-yl)butanamide
6-cyclopentyl-3-({[1-(dimethylamino)propan-2-yl]amino}methyl)-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(2,3-dimethylphenyl)-4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(2-methoxyphenyl)propanamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-hydroxyethyl)-N-(propan-2-yl)benzamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
1-(furan-2-ylmethyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
3-fluoro-N-{[4-hydroxy-1-(1-methyl-1H-imidazole-5-carbonyl)azepan-4-yl]methyl}benzamide
4-methyl-1-[4'-(2-methylpropyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl]pentane-1,2-dione
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
dimethyl({4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,3-thiazol-2-yl}methyl)amine
2-methyl-4-(piperidin-4-yl)-6-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}pyrimidine
5-chloro-2-(2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-(4-fluorophenyl)-4-(5-phenyl-1,2,4-oxadiazol-3-yl)morpholine